SCHEMBL8470432

SCHEMBL8470432

CC(CO[C]=O)c1ccc(-c2ccccc2)cc1

nearest known ligand 0.47

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
GRIA4 P48058 1/20 0.46
PTGS2 P35354 1/20 0.44
FFAR1 O14842 2/20 0.40
CHRNB2 P17787 1/20 0.39
CHRNA4 P43681 1/20 0.39
CTSS P25774 1/20 0.38
CTSK P43235 1/20 0.38
CYP1A2 P05177 1/20 0.38
GAA P10253 1/20 0.38
CYP2C9 P11712 1/20 0.38
PKM P14618 1/20 0.38
CYP2C19 P33261 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL424239 0.89 TAAR1 (0.47) FFAR1
SCHEMBL8470436 0.76 GRIA4 (0.46) GRIA4PTGS2CHRNB2CHRNA4CYP1A2
SCHEMBL2958270 0.73 APP (0.39) CYP1A2
SCHEMBL528539 0.73 CYP1A2 (0.56) GRIA4PTGS2FFAR1CYP1A2GAA
SCHEMBL20563823 0.73 CYP1A2 (0.56) GRIA4PTGS2FFAR1CYP1A2GAA
SCHEMBL6233559 0.73 KCNJ1 (0.44) CYP1A2GAA
SCHEMBL14332190 0.73 PTGS2 (0.48) GRIA4PTGS2FFAR1CHRNB2CHRNA4
SCHEMBL9572884 0.71 RIPK1 (0.47) FFAR1
SCHEMBL16687011 0.71 GRIA4 (0.51) GRIA4PTGS2CHRNB2CHRNA4
SCHEMBL1683176 0.71 CA12 (0.42) CHRNB2CHRNA4CYP1A2PKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0053540-B1 CEPHALOSPORIN DERIVATIVES AND THEIR PREPARATION RHONE-POULENC SANTE (FR) 1985-08-14 EP claimed
US-4520193-A Cephalosporin derivatives RHONE-POULENC INDUSTRIES (FR) 1985-05-28 US claimed
US-5952497-A USEFUL IN PEPTIDE, POLYPEPTIDE AND PROTEIN SYNTHESIS UNIVERSITY OF GEORGIA RESEARCH FOUNDATION (US) 1999-09-14 US disclosed
US-4520193-A Cephalosporin derivatives RHONE-POULENC INDUSTRIES (FR) 1985-05-28 US disclosed