SCHEMBL8470679

SCHEMBL8470679

Cc1c(CO)cnn1-c1ccc(Cl)cc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 1/20 0.54
CCR1 P32246 4/20 0.45
P2RX7 Q99572 2/20 0.43
NPC1 O15118 4/20 0.43
RAB9A P51151 4/20 0.43
MEN1 O00255 1/20 0.43
KMT2A Q03164 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
DRD2 P14416 3/20 0.42
DRD4 P21917 3/20 0.42
DRD3 P35462 2/20 0.42
SMN1; SMN2 Q16637 2/20 0.42
LMNA P02545 1/20 0.42
PTGS2 P35354 1/20 0.42
SMO Q99835 1/20 0.41
GRM1 Q13255 1/20 0.40
NPSR1 Q6W5P4 2/20 0.40
ALDH1A1 P00352 2/20 0.40
MAPT P10636 1/20 0.40
HSP90AA1 P07900 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4544423 0.86 SMO (0.43) NOTUMP2RX7NPC1RAB9AMEN1
SCHEMBL6532686 0.84 NPBWR1 (0.54) NOTUMP2RX7NPC1RAB9ADRD2
SCHEMBL1416762 0.83 P2RX7 (0.52) CCR1P2RX7MEN1KMT2AL3MBTL1
SCHEMBL31636507 0.83 NOTUM (0.45) NOTUMCCR1P2RX7NPC1RAB9A
SCHEMBL1568047 0.83 SMO (0.57) P2RX7NPC1RAB9ADRD2DRD4
SCHEMBL26387445 0.77 GRM1 (0.45) NOTUMCCR1NPC1RAB9AMEN1
SCHEMBL26136378 0.76 P2RX7 (0.47) NOTUMCCR1P2RX7NPC1RAB9A
SCHEMBL31636797 0.76 KMT2A (0.53) NPC1RAB9AMEN1KMT2ASMN1; SMN2
SCHEMBL5021185 0.74 NPC1 (0.45) NOTUMCCR1NPC1RAB9AMEN1
Hydrochloric Acid SCHEMBL16245892 0.72 NPC1 (0.44) NOTUMCCR1NPC1RAB9AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2014181287-A1 HETEROCYCLYL COMPOUNDS AND USES THEREOF Piramal Enterprises Limited (IN) 2014-11-13 WO disclosed
US-5990139-A 2,5-DIOXO-4-(PYRIDYL OR PHENYL-(N-HETEROCYCLE(C4N,C3N2))-ALKYLENOXY-(1,4-PHENYLENE) -)THIADIAZOLIDINES; ANTIDIABETIC AND -LIPEMIC AGENTS; SIDE EFFECT REDUCTION TAIHO PHARMACEUTICAL CO., LTD. (JP) 1999-11-23 US disclosed