SCHEMBL8474173

SCHEMBL8474173

O=C(CCl)Nc1c2c(nc3ccccc13)CCCC2

nearest known ligand 0.74

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
BCHE P06276 4/20 0.66
ACHE P22303 4/20 0.66
KDM4E B2RXH2 1/20 0.66
APP P05067 2/20 0.65
HTT P42858 2/20 0.65
GAA P10253 1/20 0.65
MAPT P10636 1/20 0.63

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9382159 0.88 KDM4E (0.65) BCHEACHEKDM4EAPPHTT
SCHEMBL9748781 0.88 KDM4E (0.68) BCHEACHEKDM4EAPPHTT
SCHEMBL9387187 0.87 KDM4E (0.69) BCHEACHEKDM4EAPPHTT
SCHEMBL9821200 0.87 BCHE (0.63) BCHEACHEAPPHTTGAA
SCHEMBL9208663 0.86 HTT (0.74) BCHEACHEKDM4EAPPHTT
SCHEMBL9384234 0.86 KDM4E (0.72) BCHEACHEKDM4EAPPHTT
SCHEMBL9232310 0.85 KDM4E (0.64) BCHEACHEKDM4EAPPHTT
SCHEMBL27524922 0.85 BCHE (0.63) BCHEACHEKDM4EAPPHTT
SCHEMBL8473136 0.85 HTT (0.69) BCHEACHEKDM4EHTTGAA
SCHEMBL9747358 0.84 KDM4E (0.63) BCHEACHEKDM4EAPPHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5861411-A TREATING DISTURBANCES OF MEMORY SUCH AS SENILE DEMENTIA AND ALZHEIMER'S DISEASE MITSUBISHI CHEMICAL CORPORATION (JP) 1999-01-19 US disclosed
EP-0746549-A1 ACETIC ACID AMIDE DERIVATIVES AND PROCESS FOR THE PREPARATION THEREOF EGIS GYOGYSZERGYAR RT. (HU) 1996-12-11 EP disclosed
US-5536728-A TREATMENT OF SENILE DEMENTIA AND ALZHEIMER'S DISEASE MITSUBISHI CHEMICAL CORPORATION (JP) 1996-07-16 US disclosed
EP-0427636-B1 4-Acylaminopyridine derivatives MITSUBISHI CHEM CORP (JP) 1996-05-29 EP disclosed
WO-1995023137-A1 ACETIC ACID AMIDE DERIVATIVES AND PROCESS FOR THE PREPARATION THEREOF EGIS Gyógyszergyár Rt. (HU) 1995-08-31 WO disclosed
US-5397785-A Activators of cholinergic neurons to treat memory disorders such as senile dementia and Alzheimer's disease MITSUBISHI KASEI CORPORATION (JP) 1995-03-14 US disclosed
EP-0319429-B1 9-Acylamino-tetrahydroacridine derivatives and memory enhancing agent containing said derivative as active ingredient MITSUBISHI CHEM IND (JP) 1994-04-27 EP disclosed
EP-0427636-A2 4-Acylaminopyridine derivatives Mitsubishi Chemical Corporation (JP) 1991-05-15 EP disclosed
US-4985430-A ALZHEIMER*S DISEASE MITSUBISHI KASEI CORPORATION (JP) 1991-01-15 US disclosed
EP-0319429-A2 9-Acylamino-tetrahydroacridine derivatives and memory enhancing agent containing said derivative as active ingredient MITSUBISHI KASEI CORPORATION (JP) 1989-06-07 EP disclosed