SCHEMBL8474456

SCHEMBL8474456

Cc1noc(-c2ccc(Cl)cc2)c1NS(=O)(=O)c1ccccc1

nearest known ligand 0.58

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
EDNRB P24530 10/20 0.58
EDNRA P25101 10/20 0.58
MAPT P10636 4/20 0.56
KDM4E B2RXH2 1/20 0.56
KDM1A O60341 1/20 0.47
TSHR P16473 1/20 0.47
MAPK1 P28482 1/20 0.47
BRD4 O60885 1/20 0.46
HSD11B1 P28845 1/20 0.46
NAT1 P18440 1/20 0.46
ALDH1A1 P00352 1/20 0.46
TP53 P04637 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8479006 0.90 EDNRB (0.60) EDNRBEDNRAMAPTKDM4ETSHR
SCHEMBL8474213 0.89 EDNRB (0.56) EDNRBEDNRATSHRMAPK1BRD4
SCHEMBL8473889 0.87 EDNRB (0.54) EDNRBEDNRAMAPTTSHRMAPK1
SCHEMBL8474221 0.86 EDNRB (0.56) EDNRBEDNRAMAPTKDM4EKDM1A
SCHEMBL14711514 0.81 LPAR1 (0.59) EDNRBEDNRAMAPTKDM4ETSHR
SCHEMBL27490281 0.81 EDNRA (0.67) EDNRBEDNRA
SCHEMBL12466034 0.80 MAPT (0.55) EDNRBEDNRAMAPTKDM4EBRD4
SCHEMBL8474683 0.79 IDH1 (0.53) EDNRBEDNRAMAPTKDM1ATSHR
SCHEMBL14790126 0.77 LPAR1 (0.50) EDNRBEDNRAMAPTKDM4ETSHR
SCHEMBL8554059 0.75 KDM1A (0.52) EDNRBEDNRAMAPTKDM4EKDM1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5859257-A ANTIINFLAMMATORY, ANTIARTHRITIC AGENTS G. D. SEARLE & CO. (US) 1999-01-12 US disclosed