SCHEMBL8475083

SCHEMBL8475083

CC(C)(C)OC(=NO)N1CCN(C(CCCC(N)=O)c2ccccc2)CC1

nearest known ligand 0.39

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 4/20 0.39
KMT2A Q03164 3/20 0.39
MEN1 O00255 2/20 0.39
C3AR1 Q16581 1/20 0.38
GLS O94925 1/20 0.37
OPRM1 P35372 5/20 0.37
OPRD1 P41143 5/20 0.37
OPRK1 P41145 5/20 0.37
OPRL1 P41146 5/20 0.37
NPSR1 Q6W5P4 1/20 0.36
CACNA1G O43497 1/20 0.35
ALDH1A1 P00352 1/20 0.34
CNR1 P21554 1/20 0.34
CNR2 P34972 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14593235 0.72 GLS (0.49) TACR1KMT2AMEN1GLSOPRD1
SCHEMBL7985622 0.70 GAA (0.50) TACR1KMT2AMEN1GLSOPRM1
SCHEMBL5410711 0.70 ATM (0.50) TACR1KMT2AMEN1GLSOPRL1
SCHEMBL8473434 0.70 GLS (0.46) TACR1KMT2AMEN1GLSALDH1A1
SCHEMBL14593385 0.68 MEN1 (0.46) TACR1KMT2AMEN1GLS
SCHEMBL4702559 0.68 GPR119 (0.50) KMT2AMEN1NPSR1ALDH1A1
SCHEMBL14593289 0.67 ABCB1 (0.51) TACR1KMT2AMEN1GLSALDH1A1
SCHEMBL14593418 0.66 MC4R (0.60) TACR1GLS
SCHEMBL4483290 0.66 SLC6A2 (0.45) KMT2AMEN1ALDH1A1CNR1CNR2
SCHEMBL28714150 0.65 GPR119 (0.50) KMT2AMEN1GLSALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5925638-A Substituted 1-indolylpropyl-4-benzylpiperazine derivatives MERCK SHARP & DOHME LTD. (GB) 1999-07-20 US disclosed
WO-1997017338-A1 SUBSTITUTED 1-INDOLYLPROPYL-4-BENZYLPIPERAZINE DERIVATIVES MERCK SHARP & DOHME LIMITED (GB) 1997-05-15 WO disclosed