SCHEMBL8475113

SCHEMBL8475113

CCCN1CC(N2CCC(c3n[nH]c4cc(F)ccc34)CC2)C(O)c2c(ccn2C)C1=O

nearest known ligand 0.37

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 13/20 0.37
HTR2A P28223 10/20 0.37
HTR1A P08908 4/20 0.37
SLC6A4 P31645 4/20 0.35
RBP4 P02753 1/20 0.32
HTR7 P34969 5/20 0.32
KCNH2 Q12809 5/20 0.32
PLK1 P53350 1/20 0.30
HTR6 P50406 1/20 0.30
MAPK1 P28482 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8473037 0.84 DRD2 (0.54) DRD2HTR2AHTR1ASLC6A4HTR7
SCHEMBL8471209 0.84 HTR1D (0.39) DRD2HTR2AHTR1ASLC6A4HTR7
SCHEMBL6773788 0.78 ADRA1D (0.41) DRD2HTR2AHTR1AHTR7KCNH2
SCHEMBL8471473 0.78 HTR2A (0.41) HTR2AHTR7
SCHEMBL8476361 0.75 CYP1A2 (0.37) DRD2HTR2AHTR1A
SCHEMBL8471130 0.75 DRD2 (0.50) DRD2HTR2AHTR1ASLC6A4HTR7
SCHEMBL8472362 0.74 DRD2 (0.54) DRD2HTR2AHTR1ASLC6A4HTR7
SCHEMBL8477450 0.74 DRD2 (0.36) DRD2HTR2AHTR1AHTR7
SCHEMBL10395172 0.72 DRD2 (0.62) DRD2HTR2ASLC6A4
SCHEMBL8471031 0.71 DRD2 (0.53) DRD2HTR2ASLC6A4HTR7KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5962448-A Pyrroloazepine derivatives SUNTORY LIMITED (JP) 1999-10-05 US disclosed