SCHEMBL8475786

SCHEMBL8475786

Cc1cc(C)cc(CN2C(=O)N(CC(=O)O)C(=O)[C@]2(C)c2ccc(C=NN)cc2)c1

nearest known ligand 0.34

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
AKR1B1 P15121 6/20 0.33
KMT2A Q03164 2/20 0.32
KDM4E B2RXH2 1/20 0.32
ALDH1A1 P00352 1/20 0.32
CYP3A4 P08684 1/20 0.32
RECQL P46063 1/20 0.32
TDP1 Q9NUW8 1/20 0.32
PTGDR2 Q9Y5Y4 3/20 0.32
LPAR1 Q92633 1/20 0.30
LPAR3 Q9UBY5 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8475817 1.00 AKR1B1 (0.33) AKR1B1KMT2AKDM4EALDH1A1CYP3A4
Hydrochloric Acid SCHEMBL6701567 0.88 ATM (0.37) AKR1B1KMT2AALDH1A1PTGDR2
SCHEMBL8481337 0.85 KMT2A (0.45) AKR1B1KMT2ACYP3A4PTGDR2
SCHEMBL8480829 0.85 KMT2A (0.45) AKR1B1KMT2ACYP3A4PTGDR2
SCHEMBL8480372 0.85 MDM2 (0.35) KMT2ARECQLPTGDR2
SCHEMBL8475358 0.85 MDM2 (0.35) KMT2ARECQLPTGDR2
SCHEMBL8523438 0.84 PTGDR2 (0.36) AKR1B1KMT2APTGDR2
Hydrochloric Acid SCHEMBL7439330 0.84 KMT2A (0.44) AKR1B1KMT2ACYP3A4PTGDR2
SCHEMBL8480629 0.84 AKR1B1 (0.42) AKR1B1
SCHEMBL7026066 0.82 ITGB3 (0.37) KMT2AKDM4EALDH1A1CYP3A4RECQL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5939556-A Hydantoin compounds, salts thereof, processes for their preparation, and processes for preparing pharmaceutically active compounds comprising them HOECHST AKTIENGESELLSCHAFT (DE) 1999-08-17 US disclosed