SCHEMBL8476183

SCHEMBL8476183

Cc1onc(-c2ccc(Cl)c(Cl)c2)c1NS(=O)(=O)c1ccccc1

nearest known ligand 0.51

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
KMO O15229 1/20 0.51
EDNRB P24530 6/20 0.48
EDNRA P25101 6/20 0.48
MT-CO2 P00403 2/20 0.47
PTGS2 P35354 2/20 0.47
ALDH1A1 P00352 2/20 0.47
NPSR1 Q6W5P4 1/20 0.47
TSHR P16473 1/20 0.47
MAPK1 P28482 1/20 0.47
PKM P14618 1/20 0.46
PTGES2 Q9H7Z7 3/20 0.44
IDH1 O75874 1/20 0.44
SLC40A1 Q9NP59 1/20 0.43
FFAR4 Q5NUL3 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8473937 0.92 IDH1 (0.48) KMOEDNRBEDNRAMT-CO2PTGS2
SCHEMBL8476626 0.88 BRD4 (0.48) EDNRBEDNRAMT-CO2PTGS2ALDH1A1
SCHEMBL8474683 0.86 IDH1 (0.53) EDNRBEDNRAMT-CO2PTGS2ALDH1A1
SCHEMBL8475736 0.85 ALDH1A1 (0.59) EDNRBEDNRAMT-CO2PTGS2ALDH1A1
SCHEMBL8475158 0.85 ALDH1A1 (0.53) EDNRBEDNRAMT-CO2PTGS2ALDH1A1
SCHEMBL6435523 0.84 ALDH1A1 (0.63) EDNRBEDNRAMT-CO2PTGS2ALDH1A1
SCHEMBL8477521 0.83 ALDH1A1 (0.58) EDNRBEDNRAMT-CO2PTGS2ALDH1A1
SCHEMBL8473536 0.83 ALDH1A1 (0.47) EDNRBEDNRAMT-CO2PTGS2ALDH1A1
SCHEMBL8477494 0.82 ALDH1A1 (0.46) EDNRBEDNRAMT-CO2PTGS2ALDH1A1
SCHEMBL8473859 0.81 PTGS2 (0.53) EDNRBEDNRAMT-CO2PTGS2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5859257-A ANTIINFLAMMATORY, ANTIARTHRITIC AGENTS G. D. SEARLE & CO. (US) 1999-01-12 US disclosed