SCHEMBL8477591

SCHEMBL8477591

CC(C(=O)CBr)N(Cc1ccccc1)Cc1ccccc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 3/20 0.51
KMT2A Q03164 3/20 0.51
HPGD P15428 2/20 0.45
NPC1 O15118 3/20 0.43
RAB9A P51151 3/20 0.43
CA12 O43570 1/20 0.43
CA9 Q16790 1/20 0.43
MMP1 P03956 2/20 0.42
MMP3 P08254 2/20 0.42
LMNA P02545 2/20 0.42
ALDH1A1 P00352 1/20 0.42
POLB P06746 1/20 0.42
HSD17B10 Q99714 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
AKT1 P31749 1/20 0.41
MMP7 P09237 1/20 0.41
MMP9 P14780 1/20 0.41
PGR P06401 1/20 0.41
ADRA2A P08913 1/20 0.41
ADRA2B P18089 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8476480 1.00 MEN1 (0.51) MEN1KMT2AHPGDNPC1RAB9A
SCHEMBL3651432 0.83 MEN1 (0.56) MEN1KMT2AHPGDNPC1RAB9A
SCHEMBL20969294 0.83 MEN1 (0.56) MEN1KMT2AHPGDNPC1RAB9A
SCHEMBL5146172 0.82 MEN1 (0.58) MEN1KMT2AHPGDNPC1RAB9A
SCHEMBL5271778 0.82 MEN1 (0.58) MEN1KMT2AHPGDNPC1RAB9A
SCHEMBL7149533 0.82 MEN1 (0.58) MEN1KMT2AHPGDNPC1RAB9A
SCHEMBL1370500 0.80 MEN1 (0.56) MEN1KMT2AHPGDNPC1RAB9A
SCHEMBL1370501 0.80 MEN1 (0.56) MEN1KMT2AHPGDNPC1RAB9A
SCHEMBL8472603 0.80 MEN1 (0.49) MEN1KMT2AHPGDNPC1RAB9A
SCHEMBL28295623 0.79 MEN1 (0.51) MEN1KMT2AHPGDNPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5990341-A Diastereoselective synthesis hydroxyethylene dipeptide isosteres EMORY UNIVERSITY (US) 1999-11-23 US disclosed
US-5587514-A Diastereoselective synthesis of hydroxyethylene dipeptide isosteres EMORY UNIVERSITY (US) 1996-12-24 US disclosed
WO-1995014655-A1 DIASTEREOSELECTIVE SYNTHESIS OF HYDROXYETHYLENE DIPEPTIDE ISOSTERES EMORY UNIVERSITY (US) 1995-06-01 WO disclosed