SCHEMBL8478332

SCHEMBL8478332

BrC/C=C/COc1ccc2c(-c3ccc(Br)cc3)coc2c1

nearest known ligand 0.69

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
LSS P48449 5/20 0.69
ALDH2 P05091 12/20 0.47
MAOA P21397 7/20 0.47
MAOB P27338 7/20 0.47
PDK1 Q15118 1/20 0.47
PDK2 Q15119 1/20 0.47
PIN1 Q13526 1/20 0.44
GSK3B P49841 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8478334 1.00 LSS (0.69) LSSALDH2MAOAMAOBPDK1
SCHEMBL4314973 0.82 LSS (1.00) LSSALDH2MAOAMAOBGSK3B
SCHEMBL4314974 0.82 LSS (1.00) LSSALDH2MAOAMAOBGSK3B
SCHEMBL30583132 0.82 LSS (1.00) LSSALDH2MAOAMAOBGSK3B
SCHEMBL8478393 0.79 ALDH2 (0.67) LSSALDH2MAOAMAOBPDK1
SCHEMBL8482529 0.77 LSS (0.69) LSS
SCHEMBL8481488 0.76 PIN1 (0.73) LSSMAOAMAOBPDK1PDK2
SCHEMBL8483516 0.76 LSS (0.69) LSS
SCHEMBL9068259 0.76 LSS (0.69) LSS
SCHEMBL25270225 0.73 ALDH2 (0.71) ALDH2MAOAMAOBPDK1PDK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5856503-A ANTICHOLESTEROL AGENTS HOFFMANN-LA ROCHE INC. (US) 1999-01-05 US disclosed
EP-0778271-A2 Aminoalkyl-substituted benzo-heterocyclic compounds F. HOFFMANN-LA ROCHE AG (CH) 1997-06-11 EP disclosed