SCHEMBL8478445

SCHEMBL8478445

Cc1cc(C)cc(C(=O)N2CCNC[C@H]2Cc2ccc(C)c(C)c2)c1

nearest known ligand 0.48

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CA1 P00915 4/20 0.48
CA2 P00918 4/20 0.48
CA4 P22748 4/20 0.48
CA9 Q16790 4/20 0.48
HCRTR1 O43613 1/20 0.47
HCRTR2 O43614 1/20 0.47
CYP3A4 P08684 1/20 0.47
TACR1 P25103 11/20 0.44
REN P00797 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL6132935 0.88 CA1 (0.46) CA1CA2CA4CA9HCRTR1
SCHEMBL7555114 0.87 CA1 (0.44) CA1CA2CA4CA9HCRTR1
SCHEMBL6132559 0.86 L3MBTL1 (0.49) CA1CA2CA4CA9HCRTR1
SCHEMBL8479516 0.86 L3MBTL1 (0.49) CA1CA2CA4CA9HCRTR1
SCHEMBL9242103 0.86 L3MBTL1 (0.49) CA1CA2CA4CA9HCRTR1
SCHEMBL8480340 0.86 CA1 (0.64) CA1CA2CA4CA9HCRTR1
SCHEMBL7555118 0.85 CA1 (0.44) CA1CA2CA4CA9HCRTR1
Hydrochloric Acid SCHEMBL9240138 0.85 L3MBTL1 (0.48) CA1CA2CA4CA9HCRTR1
Hydrochloric Acid SCHEMBL8476515 0.85 L3MBTL1 (0.48) CA1CA2CA4CA9HCRTR1
Fumaric Acid SCHEMBL7554500 0.81 TACR1 (0.46) CA1CA2CA4CA9HCRTR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5883098-A USED AS TACHYKININ ANTAGONISTS IN THE TREATMENT OF RESPIRATORY DISEASES, OPHTHALMIC DISEASES AND INFLAMMATORY DISEASES FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1999-03-16 US disclosed
US-5670505-A TACHYKIKIN ANTAGONIST FOR RESPIRATORY DISEASES, OPHTHALMIC DISEASES AND ANTIINFLAMMATORY AGENTS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1997-09-23 US disclosed
EP-0655442-A1 Piperazine derivatives as Tachykinin antagonists FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1995-05-31 EP disclosed