SCHEMBL8480171

SCHEMBL8480171

Cc1cc(C)c(-c2nc(-c3ccccn3)c(-c3ccc(F)cc3)[nH]2)c(C)c1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TGFBR1 P36897 1/20 0.48
MAPK14 Q16539 9/20 0.47
MAPK13 O15264 6/20 0.47
GCGR P47871 6/20 0.47
MAPK12 P53778 6/20 0.47
MAPK11 Q15759 6/20 0.47
CSNK1D P48730 4/20 0.46
CSNK1E P49674 3/20 0.46
ALOX5 P09917 4/20 0.46
METAP2 P50579 2/20 0.43
METAP1 P53582 2/20 0.43
CBFB Q13951 2/20 0.43
PRKD3 O94806 1/20 0.43
MAP4K4 O95819 1/20 0.43
FRK P42685 1/20 0.43
MAPK9 P45984 1/20 0.43
CSNK1A1 P48729 1/20 0.43
GSK3B P49841 1/20 0.43
PTK6 Q13882 1/20 0.43
PRKD2 Q9BZL6 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8475950 0.88 MAPK14 (0.45) MAPK14MAPK13GCGRMAPK12MAPK11
SCHEMBL8480160 0.85 MAPK14 (0.49) TGFBR1MAPK14MAPK13GCGRMAPK12
SCHEMBL8479495 0.85 MAPK14 (0.49) TGFBR1MAPK14CSNK1DCSNK1EMETAP2
SCHEMBL6960991 0.81 MAPK14 (0.72) MAPK14MAPK13GCGRMAPK12MAPK11
SCHEMBL5921871 0.81 MAPK14 (0.72) MAPK14MAPK13GCGRMAPK12MAPK11
SCHEMBL8476402 0.79 MAPK13 (0.47) MAPK14MAPK13GCGRMAPK12MAPK11
SCHEMBL4526549 0.76 TGFBR1 (0.53) TGFBR1MAPK14MAPK13GCGRMAPK12
SCHEMBL5623031 0.76 KDM4E (0.57) MAPK14MAPK13GCGRMAPK12MAPK11
SCHEMBL8481652 0.74 MAPK13 (0.43) MAPK14MAPK13GCGRMAPK12MAPK11
SCHEMBL8480021 0.74 MAPK13 (0.44) MAPK14MAPK13GCGRMAPK12MAPK11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5959113-A REACTING A DIKETONE DERIVATIVE WITH AN ALDEHYDE DERIVATIVE; ADMINISTERING TO TREAT ATHEROSCLEROSIS, PSORIASIS, ALOPECIA AND TUMORS HOFFMANN-LA ROCHE INC. (US) 1999-09-28 US claimed
US-5959113-A REACTING A DIKETONE DERIVATIVE WITH AN ALDEHYDE DERIVATIVE; ADMINISTERING TO TREAT ATHEROSCLEROSIS, PSORIASIS, ALOPECIA AND TUMORS HOFFMANN-LA ROCHE INC. (US) 1999-09-28 US disclosed