SCHEMBL8480279

SCHEMBL8480279

COCOc1ccc(N2CCCCC2)c(F)c1-c1ccc(C(=O)O)c(C)c1O

nearest known ligand 0.38

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
MRGPRX4 Q96LA9 2/20 0.38
ERAP1 Q9NZ08 2/20 0.34
ALDH1A1 P00352 2/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
MAPT P10636 1/20 0.33
HPGD P15428 1/20 0.33
TSHR P16473 1/20 0.33
RARA P10276 1/20 0.33
RARB P10826 1/20 0.33
RARG P13631 1/20 0.33
KDM4E B2RXH2 1/20 0.32
ABCC8 Q09428 1/20 0.32
F11 P03951 2/20 0.32
GAA P10253 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
F2 P00734 1/20 0.32
KLKB1 P03952 1/20 0.32
NPC1 O15118 1/20 0.32
RAB9A P51151 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8479739 0.99 MRGPRX4 (0.39) MRGPRX4ERAP1MAPTRARARARB
SCHEMBL8481719 0.83 MAPT (0.41) MAPT
SCHEMBL8478791 0.83 EGFR (0.36)
SCHEMBL8480273 0.79 MRGPRX4 (0.41) MRGPRX4ERAP1ALDH1A1SMN1; SMN2MAPT
SCHEMBL8479735 0.78 MRGPRX4 (0.41) MRGPRX4ERAP1MAPTRARARARB
SCHEMBL8477001 0.74 EGFR (0.37) ALDH1A1HPGDKDM4E
SCHEMBL8480189 0.73 ERAP1 (0.46) ERAP1ALDH1A1SMN1; SMN2MAPTHPGD
SCHEMBL8476017 0.72 ERAP1 (0.44) ERAP1ALDH1A1MAPTHPGDTSHR
SCHEMBL8480277 0.69 ERAP1 (0.40) ERAP1ALDH1A1SMN1; SMN2MAPTHPGD
SCHEMBL6215857 0.69 ALDH1A1 (0.44) ERAP1ALDH1A1SMN1; SMN2MAPTHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5914406-A ENZYME INHIBITOR; USEFUL FOR TREATMENT OF INFLAMMATORY SKIN DISORDERS AND ALOPECIA HOFFMAN-LA ROCHE INC. (US) 1999-06-22 US disclosed
US-5750706-A TREATMENT OF INFLAMMATORY SKIN DISORDERS AND ALOPECIA HOFFMANN-LA ROCHE INC. (US) 1998-05-12 US disclosed