SCHEMBL8480439

SCHEMBL8480439

O=S(=O)(c1ccccc1)n1cc(-c2cn[nH]c2)c2cc(CC3=CCCC3)cnc21

nearest known ligand 0.35

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HTR6 P50406 9/20 0.35
BRD4 O60885 3/20 0.34
PDPK1 O15530 2/20 0.34
CHUK O15111 2/20 0.33
CA12 O43570 1/20 0.33
CA9 Q16790 1/20 0.33
BCL2L1 Q07817 1/20 0.33
GRK2 P25098 1/20 0.33
PTPN11 Q06124 1/20 0.32
DRD2 P14416 1/20 0.32
HTR2A P28223 1/20 0.32
HTR7 P34969 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8443783 0.86 BCL2L1 (0.41) HTR6BRD4CHUKCA12CA9
SCHEMBL3354967 0.85 PDPK1 (0.40) HTR6BRD4PDPK1PTPN11
SCHEMBL8480893 0.80 BRD4 (0.38) HTR6BRD4PDPK1CHUKCA12
SCHEMBL8443973 0.79 SCN9A (0.39) HTR6BRD4PDPK1CHUKCA12
SCHEMBL2752527 0.77 HTR6 (0.41) HTR6BRD4PDPK1CHUKCA12
SCHEMBL8443781 0.77 BRD4 (0.44) HTR6BRD4PDPK1CHUKCA12
SCHEMBL16374479 0.77 BRD4 (0.43) HTR6BRD4PDPK1CHUKCA12
SCHEMBL3348977 0.76 HTR6 (0.48) HTR6BRD4DRD2HTR2AHTR7
SCHEMBL16374566 0.76 ROCK2 (0.40) HTR6BRD4CHUKCA12CA9
SCHEMBL8169943 0.76 ROCK2 (0.40) HTR6BRD4CHUKCA12CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1749829-B1 JNK inhibitors EISAI R&D MAN CO LTD (JP) 2010-11-03 EP disclosed