SCHEMBL8480469

SCHEMBL8480469

CCOC(=O)c1ccc(C2=NNC(=O)C(C)C2)cc1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 2/20 0.59
RAB9A P51151 4/20 0.58
PDE3B Q13370 2/20 0.48
PDE3A Q14432 2/20 0.48
HRH3 Q9Y5N1 1/20 0.47
KDM4E B2RXH2 2/20 0.44
CA12 O43570 1/20 0.43
CA1 P00915 1/20 0.43
CA2 P00918 1/20 0.43
ESR1 P03372 1/20 0.43
CA7 P43166 1/20 0.43
CA9 Q16790 1/20 0.43
ESR2 Q92731 1/20 0.43
CA14 Q9ULX7 1/20 0.43
ALDH1A1 P00352 4/20 0.43
MAPT P10636 3/20 0.43
SMN1; SMN2 Q16637 3/20 0.43
NR3C2 P08235 1/20 0.43
MEN1 O00255 1/20 0.43
KMT2A Q03164 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8481664 0.78 LMNA (0.56) LMNARAB9APDE3BPDE3AHRH3
SCHEMBL9659827 0.77 PDE3B (0.58) LMNARAB9APDE3BPDE3AHRH3
SCHEMBL7277682 0.74 LMNA (0.78) LMNARAB9APDE3BPDE3AKDM4E
SCHEMBL28802880 0.74 LMNA (1.00) LMNARAB9AALDH1A1MAPTSMN1; SMN2
SCHEMBL7264498 0.74 PDE3B (0.58) LMNARAB9APDE3BPDE3AHRH3
SCHEMBL1754736 0.73 GPR119 (0.61) LMNARAB9APDE3BPDE3AHRH3
SCHEMBL11400199 0.73 MAPT (0.57) LMNARAB9APDE3BPDE3AHRH3
SCHEMBL7272078 0.73 PDE3B (0.64) LMNARAB9APDE3BPDE3AHRH3
SCHEMBL16351874 0.71 CA1 (0.73) LMNARAB9AKDM4ECA12CA1
SCHEMBL1965326 0.71 CA1 (0.73) LMNARAB9AKDM4ECA12CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5883090-A Endothelin receptor antagonists MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1999-03-16 US disclosed