SCHEMBL8480828

SCHEMBL8480828

CCS(=O)(=O)CCC(NC1CC(C)(C)Oc2ccc(F)cc21)C(=O)O

nearest known ligand 0.47

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
TRPV1 Q8NER1 15/20 0.47
CYP3A4 P08684 1/20 0.42
KCNE1 P15382 3/20 0.41
KCNQ1 P51787 3/20 0.41
CTSD P07339 2/20 0.40
BACE1 P56817 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8476969 0.84 TRPV1 (0.36) TRPV1CTSDBACE1
SCHEMBL8480422 0.82 TRPV1 (0.50) TRPV1CYP3A4KCNE1KCNQ1CTSD
SCHEMBL8482068 0.81 TSHR (0.42) TRPV1CYP3A4
SCHEMBL6558672 0.78 TRPV1 (0.49) TRPV1CYP3A4KCNE1KCNQ1CTSD
SCHEMBL8477265 0.77 TRPV1 (0.49) TRPV1CYP3A4KCNE1KCNQ1CTSD
SCHEMBL8476718 0.77 TRPV1 (0.38) TRPV1CTSDBACE1
SCHEMBL6560804 0.76 TRPV1 (0.48) TRPV1CYP3A4KCNE1KCNQ1CTSD
SCHEMBL7828519 0.75 TRPV1 (0.45) TRPV1CYP3A4KCNE1KCNQ1CTSD
SCHEMBL6559589 0.74 TRPV1 (0.52) TRPV1CYP3A4KCNE1KCNQ1
Guanidine SCHEMBL8525006 0.73 TRPV1 (0.35) TRPV1CTSDBACE1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5955607-A TREATING CARDIOVASCULAR AND GASTROINTESTINAL DISORDERS HOECHST MARION ROUSSEL DEUTSCHLAND (DE) 1999-09-21 US disclosed