SCHEMBL8480921

SCHEMBL8480921

Cc1[c]cc(-c2ccccc2)c(-c2ccccc2)c1C

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDCD1 Q15116 1/20 0.36
CD274 Q9NZQ7 1/20 0.36
CYP2A6 P11509 1/20 0.35
CYP2B6 P20813 1/20 0.35
KMT2A Q03164 2/20 0.35
MEN1 O00255 1/20 0.35
NPC1 O15118 1/20 0.35
RAB9A P51151 1/20 0.35
AKT2 P31751 3/20 0.33
BRD4 O60885 2/20 0.33
CHEK1 O14757 1/20 0.33
AKT1 P31749 1/20 0.33
BRD2 P25440 1/20 0.33
ESR2 Q92731 1/20 0.33
LMNA P02545 1/20 0.33
MAPT P10636 1/20 0.33
HTT P42858 1/20 0.33
SQOR Q9Y6N5 1/20 0.33
PTGS1 P23219 1/20 0.32
PTGS2 P35354 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12816030 0.86 CYP2A6 (0.36) PDCD1CD274CYP2A6CYP2B6KMT2A
SCHEMBL8482076 0.84 ACHE (0.32) PTGS1PTGS2
SCHEMBL9412187 0.83 PDCD1 (0.38) PDCD1CD274CYP2A6CYP2B6AKT2
SCHEMBL11722877 0.82 MAPT (0.34) CYP2A6CYP2B6KMT2AMEN1NPC1
SCHEMBL8479313 0.78 PDE4B (0.45) KMT2AMEN1NPC1RAB9AMAPT
SCHEMBL5188189 0.78 HPRT1 (0.37) KMT2AMEN1NPC1RAB9ALMNA
SCHEMBL8476959 0.78 PDCD1 (0.36) PDCD1CD274CYP2A6CYP2B6KMT2A
SCHEMBL8477304 0.75 PDCD1 (0.38) PDCD1CD274CYP2A6CYP2B6KMT2A
SCHEMBL8474110 0.75 GCGR (0.35) PDCD1CD274CYP2A6CYP2B6KMT2A
SCHEMBL7385531 0.73 CYP2A6 (0.38) PDCD1CD274CYP2A6CYP2B6KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8937195-B2 Method for producing the transition metal complex, catalyst for trimerization, method for producing 1-hexene, method for producing the substituted cyclopentadiene compound (1) SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 2015-01-20 US disclosed
EP-2691406-A1 METHOD FOR PRODUCING THE TRANSITION METAL COMPLEX, CATALYST FOR TRIMERIZATION, METHOD FOR PRODUCING 1-HEXENE, METHOD FOR PRODUCING THE SUBSTITUTED CYCLOPENTADIENE COMPOUND (1) Sumitomo Chemical Company, Limited (JP) 2014-02-05 EP disclosed
US-20140018564-A1 METHOD FOR PRODUCING THE TRANSITION METAL COMPLEX, CATALYST FOR TRIMERIZATION, METHOD FOR PRODUCING 1-HEXENE, METHOD FOR PRODUCING THE SUBSTITUTED CYCLOPENTADIENE COMPOUND (1) SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 2014-01-16 US disclosed
WO-2012133935-A1 METHOD FOR PRODUCING THE TRANSITION METAL COMPLEX, CATALYST FOR TRIMERIZATION, METHOD FOR PRODUCING 1-HEXENE, METHOD FOR PRODUCING THE SUBSTITUTED CYCLOPENTADIENE COMPOUND (3) SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 2012-10-04 WO disclosed
WO-2012133924-A1 METHOD FOR PRODUCING THE TRANSITION METAL COMPLEX, CATALYST FOR TRIMERIZATION, METHOD FOR PRODUCING 1-HEXENE, METHOD FOR PRODUCING THE SUBSTITUTED CYCLOPENTADIENE COMPOUND (1) SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 2012-10-04 WO disclosed
US-6004988-A Carboxylic acid derivatives, their preparation and their use BASF AKTIENGESELLSCHAFT (DE) 1999-12-21 US disclosed
US-4361707-A COBALT, IODINE AND A PHOSPHINE LIGAND GULF RESEARCH & DEVELOPMENT COMPANY (US) 1982-11-30 US disclosed