SCHEMBL8480988

SCHEMBL8480988

COc1ccc(-c2cccc(Cl)c2)cc1

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABL1 P00519 2/20 0.63
ABCB1 P08183 2/20 0.63
BCR P11274 2/20 0.63
RELA Q04206 1/20 0.56
KMT2A Q03164 1/20 0.55
HDAC4 P56524 1/20 0.54
HDAC2 Q92769 1/20 0.54
HDAC8 Q9BY41 1/20 0.54
TAAR1 Q96RJ0 2/20 0.53
ALOX5 P09917 2/20 0.50
CYP1A1 P04798 1/20 0.50
CYP1A2 P05177 1/20 0.50
CYP2E1 P05181 1/20 0.50
CYP3A4 P08684 1/20 0.50
CYP2C8 P10632 1/20 0.50
CYP2D6 P10635 1/20 0.50
CYP2A6 P11509 1/20 0.50
CYP2C9 P11712 1/20 0.50
CYP4B1 P13584 1/20 0.50
CYP2B6 P20813 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30996183 1.00 ABL1 (0.63) ABL1ABCB1BCRRELAKMT2A
SCHEMBL792094 0.86 CYP1A1 (0.57) ABL1ABCB1BCRRELAHDAC4
SCHEMBL1180429 0.85 ABL1 (0.83) ABL1ABCB1BCRHDAC4HDAC2
SCHEMBL16394285 0.82 TAAR1 (0.71) TAAR1ALOX5CYP1A2ESR2BACE1
SCHEMBL31491189 0.82 TAAR1 (0.71) TAAR1ALOX5CYP1A2ESR2BACE1
SCHEMBL792197 0.81 ABL1 (0.77) ABL1ABCB1BCRHDAC4HDAC2
SCHEMBL27649742 0.81 ABL1 (0.77) ABL1ABCB1BCRKMT2AHDAC4
SCHEMBL1180412 0.81 ABL1 (0.77) ABL1ABCB1BCRHDAC4HDAC2
SCHEMBL20669453 0.80 TAAR1 (0.68) KMT2ATAAR1ALOX5CYP1A2ESR2
SCHEMBL6314185 0.80 KMT2A (0.46) ABL1ABCB1BCRRELAKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3674303-B1 NOVEL TRYPTOPHAN HYDROXYLASE INHIBITOR AND PHARMACEUTICAL COMPOSITION INCLUDING SAME GWANGJU INST SCIENCE & TECH (KR) 2022-07-20 EP claimed
CN-104892539-B Novel synthesis method of iron-catalyzed 2-aryl benzoxazole compound 苏州大学 2017-12-22 CN disclosed
US-20100144516-A1 PREPARATION AND USE OF MAGNESIUM AMIDES LUDWIG-MAXIMILIANS-UNIVERSITAT MUNCHEN (DE) 2010-06-10 US disclosed
US-20100144516-A1 PREPARATION AND USE OF MAGNESIUM AMIDES LUDWIG-MAXIMILIANS-UNIVERSITAT MUNCHEN (DE) 2010-06-10 US disclosed
WO-2008087057-A1 PREPARATION AND USE OF MAGNESIUM AMIDES LUDWIG-MAXIMILIANS-UNIVERSITAET MUENCHEN (DE) 2008-07-24 WO disclosed
US-5977105-A Compounds ASTRA PHARMAEUTICALS LTD. (GB) 1999-11-02 US disclosed
EP-0865431-A2 COMPOUNDS Astra Pharmaceuticals Limited (GB) 1998-09-23 EP disclosed
WO-1997020815-A1 COMPOUNDS ASTRA PHARMACEUTICALS LTD. (GB) 1997-06-12 WO disclosed