SCHEMBL8481963

SCHEMBL8481963

CCS(=O)(=O)C(NC1CC(C)(C)Oc2ccc(F)cc21)C(=O)NCCc1ccccn1

nearest known ligand 0.44

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
TRPV1 Q8NER1 13/20 0.44
CYP3A4 P08684 2/20 0.42
HTT P42858 2/20 0.40
ATM Q13315 1/20 0.40
TSHR P16473 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
HSD11B1 P28845 1/20 0.38
RAB9A P51151 1/20 0.37
MME P08473 1/20 0.37
ECE1 P42892 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8476611 0.88 TRPV1 (0.49) TRPV1CYP3A4HTT
SCHEMBL8482068 0.86 TSHR (0.42) TRPV1CYP3A4HTTATMTSHR
SCHEMBL8482576 0.85 TRPV1 (0.49) TRPV1CYP3A4
SCHEMBL8480649 0.80 TRPV1 (0.47) TRPV1CYP3A4
SCHEMBL8481888 0.80 TRPV1 (0.50) TRPV1CYP3A4
SCHEMBL8477642 0.79 TRPV1 (0.42) TRPV1CYP3A4HTTATMSMN1; SMN2
SCHEMBL8480422 0.79 TRPV1 (0.50) TRPV1CYP3A4
SCHEMBL8476363 0.79 TRPV1 (0.47) TRPV1CYP3A4
SCHEMBL8477265 0.79 TRPV1 (0.49) TRPV1CYP3A4
SCHEMBL8481389 0.78 TRPV1 (0.44) TRPV1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5955607-A TREATING CARDIOVASCULAR AND GASTROINTESTINAL DISORDERS HOECHST MARION ROUSSEL DEUTSCHLAND (DE) 1999-09-21 US disclosed