SCHEMBL8482120

SCHEMBL8482120

COc1ccccc1N1CCc2c1c1cccc(C)c1[nH]c2=O

nearest known ligand 0.85

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.57
ALDH1A1 P00352 1/20 0.57
GLA P06280 1/20 0.44
GAA P10253 1/20 0.44
HTT P42858 1/20 0.44
TNKS O95271 2/20 0.43
TNKS2 Q9H2K2 2/20 0.43
PARP10 Q53GL7 1/20 0.43
PARP2 Q9UGN5 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8487682 0.92 KDM4E (0.58) KDM4EALDH1A1GLAGAAHTT
SCHEMBL8484042 0.91 KDM4E (0.52) KDM4EALDH1A1
SCHEMBL9686536 0.88 DDB1 (0.48) KDM4E
SCHEMBL9685709 0.86 KDM4E (0.46) KDM4EALDH1A1TNKSTNKS2PARP10
SCHEMBL7498546 0.85 KDM4E (0.51) KDM4EALDH1A1GLAGAAHTT
SCHEMBL7495661 0.83 KDM4E (0.48) KDM4EALDH1A1GLAGAAHTT
SCHEMBL8481514 0.83 CYP1A2 (0.43) GAA
SCHEMBL8484525 0.81 NQO2 (0.44) KDM4EALDH1A1GLAGAAHTT
SCHEMBL8487677 0.81 CYP1A2 (0.46) KDM4EALDH1A1GAA
SCHEMBL8071575 0.81 KDM4E (0.41) KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5914402-A Process for preparing 1-aryl-4-oxopyrrolo 3,2-c! quinoline derivatives KOREA RESEARCH INSTITUTE OF CHEMICAL TECHNOLOGY (KR) 1999-06-22 US disclosed