SCHEMBL9685709

SCHEMBL9685709

COc1cccc2c3c(c(=O)[nH]c12)CCCN3c1ccccc1C

nearest known ligand 0.76

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.46
ALDH1A1 P00352 1/20 0.46
HPGD P15428 1/20 0.45
NQO2 P16083 1/20 0.43
TNKS O95271 2/20 0.43
TNKS2 Q9H2K2 2/20 0.43
PARP10 Q53GL7 1/20 0.43
PARP2 Q9UGN5 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8484042 0.94 KDM4E (0.52) KDM4EALDH1A1HPGD
SCHEMBL8487682 0.86 KDM4E (0.58) KDM4EALDH1A1HPGDTNKSTNKS2
SCHEMBL8482120 0.86 KDM4E (0.57) KDM4EALDH1A1TNKSTNKS2PARP10
SCHEMBL9686536 0.83 DDB1 (0.48) KDM4E
SCHEMBL8071575 0.82 KDM4E (0.41) KDM4EALDH1A1
SCHEMBL8487677 0.82 CYP1A2 (0.46) KDM4EALDH1A1HPGDNQO2
SCHEMBL8484525 0.82 NQO2 (0.44) KDM4EALDH1A1HPGDNQO2
SCHEMBL7488966 0.80 ADRA1D (0.42) KDM4EALDH1A1
SCHEMBL8480746 0.80 KDM4E (0.58) KDM4EALDH1A1HPGDNQO2
SCHEMBL8066947 0.78 KDM4E (0.38) KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0307078-B1 QUINOLINE DERIVATIVES, PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM SMITHKLINE BEECHAM INTERCREDIT B.V. (NL) 1992-08-26 EP disclosed
US-5051508-A Antisecretory agents and enzyme inhibitors as antiulcer agents SMITHKLINE BECKMAN INTERCREDIT B.V. (NL) 1991-09-24 US disclosed
EP-0307078-A1 Quinoline derivatives, process for their preparation and pharmaceutical compositions containing them SMITHKLINE BEECHAM INTERCREDIT B.V. (NL) 1989-03-15 EP disclosed