SCHEMBL8484401

SCHEMBL8484401

Cc1cc(C)c(Nc2cc(Cl)nc(C)n2)c(C)c1

nearest known ligand 0.49

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
RAPGEF4 Q8WZA2 13/20 0.48
CRHR1 P34998 2/20 0.45
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41
NPC1 O15118 1/20 0.40
RAB9A P51151 1/20 0.40
POLB P06746 1/20 0.40
GAA P10253 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1183306 0.86 RAPGEF4 (0.48) RAPGEF4
SCHEMBL1193784 0.83 MAPT (0.50) RAPGEF4KMT2ANPC1RAB9APOLB
SCHEMBL7068369 0.79 RAPGEF4 (0.48) RAPGEF4CRHR1
SCHEMBL4857708 0.79 CRHR1 (0.49) RAPGEF4CRHR1MEN1KMT2ANPC1
SCHEMBL10303879 0.78 RAPGEF4 (0.64) RAPGEF4
SCHEMBL18971579 0.77 CHRNA7 (0.47) MEN1KMT2ANPC1RAB9APOLB
SCHEMBL29849205 0.72 MEN1 (0.47) MEN1KMT2ANPC1RAB9APOLB
SCHEMBL3711167 0.72 MEN1 (0.47) MEN1KMT2ANPC1RAB9APOLB
SCHEMBL1183435 0.72 RAPGEF4 (0.45) RAPGEF4
SCHEMBL6093823 0.72 CRHR1 (0.43) RAPGEF4CRHR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5962479-A Corticotropin releasing factor antagonists PFIZER INC. (US) 1999-10-05 US disclosed