SCHEMBL8484497

SCHEMBL8484497

c1ccc(CN2CCC(n3nnc(-c4ccccc4)n3)CC2)cc1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
DRD4 P21917 13/20 1.00
DRD2 P14416 12/20 1.00
DRD3 P35462 11/20 1.00
RAB9A P51151 1/20 0.54
L3MBTL1 Q9Y468 1/20 0.54
KCNH2 Q12809 2/20 0.51
SIGMAR1 Q99720 1/20 0.51
KMT2A Q03164 2/20 0.50
MEN1 O00255 1/20 0.50
SMN1; SMN2 Q16637 1/20 0.49
LMNA P02545 1/20 0.49
MAPT P10636 1/20 0.49
NTSR1 P30989 1/20 0.49
HTT P42858 1/20 0.49
NPSR1 Q6W5P4 1/20 0.49
CYP2D6 P10635 1/20 0.48
ACHE P22303 1/20 0.48
CCR3 P51677 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20816392 0.78 DRD2 (0.63) DRD4DRD2DRD3RAB9AL3MBTL1
SCHEMBL4959931 0.77 DRD2 (0.62) DRD4DRD2DRD3RAB9AL3MBTL1
SCHEMBL4319291 0.76 DRD2 (0.60) DRD4DRD2DRD3RAB9AL3MBTL1
SCHEMBL8482373 0.73 DRD4 (1.00) DRD4DRD2DRD3KCNH2SIGMAR1
SCHEMBL9278989 0.73 DRD4 (1.00) DRD4DRD2DRD3KCNH2SIGMAR1
Hydrochloric Acid SCHEMBL8482360 0.72 DRD4 (0.97) DRD4DRD2DRD3KCNH2SIGMAR1
SCHEMBL8484877 0.71 DRD4 (1.00) DRD4DRD2DRD3KCNH2SIGMAR1
SCHEMBL8482378 0.71 DRD4 (1.00) DRD4DRD2DRD3KCNH2SIGMAR1
SCHEMBL2359215 0.71 DRD2 (0.55) DRD4DRD2DRD3RAB9AL3MBTL1
SCHEMBL4413466 0.71 RAB9A (1.00) RAB9AL3MBTL1KMT2ASMN1; SMN2LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1996021660-A1 FIVE-MEMBERED HETEROAROMATIC COMPOUNDS AS DOPAMINE RECEPTOR SUBTYPE LIGANDS MERCK SHARP & DOHME LIMITED (GB) 1996-07-18 WO claimed
US-5939436-A Five-membered heteroaromatic compounds as dopamine receptor subtype ligands MERCK SHARP & DOHME LTD. (GB) 1999-08-17 US disclosed
WO-1996021660-A1 FIVE-MEMBERED HETEROAROMATIC COMPOUNDS AS DOPAMINE RECEPTOR SUBTYPE LIGANDS MERCK SHARP & DOHME LIMITED (GB) 1996-07-18 WO disclosed