SCHEMBL8486271

SCHEMBL8486271

CCOc1cccc2c(C)c(C(N)=O)oc12

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 7/20 0.53
ALDH1A1 P00352 4/20 0.53
HPGD P15428 4/20 0.53
L3MBTL1 Q9Y468 3/20 0.53
HSD17B10 Q99714 1/20 0.53
MCL1 Q07820 1/20 0.46
CYP1A2 P05177 1/20 0.44
CYP3A4 P08684 1/20 0.44
CYP2C19 P33261 1/20 0.44
MAPK10 P53779 2/20 0.42
TDP1 Q9NUW8 2/20 0.41
AHR P35869 1/20 0.41
MAPT P10636 2/20 0.40
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
PABPC1 P11940 1/20 0.40
CYP2A6 P11509 1/20 0.40
CA12 O43570 1/20 0.40
CA1 P00915 1/20 0.40
CA2 P00918 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13699676 0.86 CYP1A2 (0.44) KDM4EALDH1A1HPGDL3MBTL1HSD17B10
SCHEMBL8509407 0.86 KDM4E (0.53) KDM4EALDH1A1HPGDL3MBTL1HSD17B10
Hydrochloric Acid SCHEMBL8483294 0.83 KDM4E (0.44) KDM4EALDH1A1HPGDL3MBTL1HSD17B10
SCHEMBL11233136 0.78 ATM (0.54) KDM4EHPGDL3MBTL1MCL1TDP1
SCHEMBL13699889 0.78 TP53 (0.60) KDM4EALDH1A1HPGDHSD17B10CYP1A2
SCHEMBL13699726 0.76 MAPT (0.53) KDM4EALDH1A1HPGDL3MBTL1HSD17B10
SCHEMBL8119758 0.76 KMT2A (0.49) KDM4EALDH1A1CYP1A2CYP3A4CYP2C19
SCHEMBL13699704 0.75 MAPT (0.60) ALDH1A1HPGDHSD17B10MAPK10AHR
SCHEMBL73391 0.75 KDM4E (0.52) KDM4EALDH1A1HPGDL3MBTL1HSD17B10
SCHEMBL4745049 0.75 RAB9A (0.56) KDM4EHPGDL3MBTL1MCL1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5955495-A BENZOFURAN-2-CARBOXAMIDINE OR 2-CARBOXAMIDOXIME COMPOUNDS USEFUL IN THE CONTROL OR PREVENTION OF ILLNESSES OR DISORDERS OF THE CENTRAL NERVOUS SYSTEM SUCH AS MIGRAINE, SCHIZOPHRENIA, ANXIETY STATES, SLEEP DISORDERS, ANOREXIA, ALZHEIMER'S HOFFMANN-LA ROCHE INC. (US) 1999-09-21 US disclosed
EP-0906301-A1 BENZOFURYL DERIVATIVES AND THEIR USE F. HOFFMANN-LA ROCHE AG (CH) 1999-04-07 EP disclosed
WO-1997042183-A1 BENZOFURYL DERIVATIVES AND THEIR USE F. HOFFMANN-LA ROCHE AG (CH) 1997-11-13 WO disclosed