SCHEMBL8487679

SCHEMBL8487679

CCOC(=O)C(c1ccc(Br)s1)C1CCCCCC1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 4/20 0.43
ALDH1A1 P00352 4/20 0.42
GAA P10253 2/20 0.42
KMT2A Q03164 2/20 0.42
SLC6A2 P23975 5/20 0.42
SLC6A3 Q01959 5/20 0.42
CYP3A4 P08684 2/20 0.42
CHRM2 P08172 1/20 0.42
HTR1A P08908 1/20 0.42
ADRA2A P08913 1/20 0.42
CHRM1 P11229 1/20 0.42
DRD1 P21728 1/20 0.42
ADRA1A P35348 1/20 0.42
OPRM1 P35372 1/20 0.42
DRD3 P35462 1/20 0.42
KCNH2 Q12809 1/20 0.42
LMNA P02545 1/20 0.42
CYP1A2 P05177 1/20 0.42
CYP2D6 P10635 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4240183 0.81 KDM4E (0.41) TSHRALDH1A1GAAKMT2ASLC6A2
SCHEMBL8486695 0.77 TSHR (0.47) TSHRALDH1A1GAAKMT2ASLC6A2
SCHEMBL4245904 0.76 SLC6A2 (0.45) TSHRALDH1A1KMT2ASLC6A2SLC6A3
SCHEMBL11932077 0.75 SLC6A3 (0.51) TSHRGAAKMT2ASLC6A2SLC6A3
SCHEMBL1164590 0.74 POLB (0.41) TSHRALDH1A1GAAKMT2ALMNA
SCHEMBL10955574 0.73 SLC6A2 (0.70) TSHRKMT2ASLC6A2SLC6A3CYP3A4
SCHEMBL11366829 0.72 SLC6A3 (0.48) TSHRALDH1A1GAAKMT2ASLC6A2
SCHEMBL28632940 0.72 SLC6A2 (0.67) TSHRKMT2ASLC6A2SLC6A3CYP3A4
SCHEMBL6951792 0.70 TSHR (0.51) TSHRALDH1A1GAAKMT2ASLC6A2
SCHEMBL14862650 0.70 SLC6A3 (0.46) TSHRALDH1A1SLC6A2SLC6A3CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5925646-A Heterocyclic aryl-, alkyl- and cycloalkylacetamides BAYER AKTIENGESELLSCHAFT (DE) 1999-07-20 US disclosed
US-5747505-A Heterocyclic aryl-, alkyl- and cycloalkylacetamides BAYER AKTIENGESELLSCHAFT (DE) 1998-05-05 US disclosed