SCHEMBL8488703

SCHEMBL8488703

CS(=O)(=O)c1nccc(-n2cc(-c3cccc(C(F)(F)F)c3)nc2C2CCCCN2C(=O)OCc2ccccc2)n1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BTK Q06187 2/20 0.41
TMEM97 Q5BJF2 5/20 0.40
SIGMAR1 Q99720 5/20 0.40
CPT2 P23786 3/20 0.39
CPT1A P50416 3/20 0.39
CPT1B Q92523 2/20 0.39
AADAT Q8N5Z0 2/20 0.37
CNR2 P34972 2/20 0.36
RORC P51449 1/20 0.36
F2R P25116 1/20 0.36
ALDH1A1 P00352 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
TRPV1 Q8NER1 1/20 0.35
EGFR P00533 1/20 0.35
CYP3A4 P08684 1/20 0.35
BRAF P15056 1/20 0.35
JAK3 P52333 1/20 0.35
MAPK10 P53779 1/20 0.35
KCNH2 Q12809 1/20 0.35
ERBB4 Q15303 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8487384 0.86 BTK (0.45) BTKTMEM97SIGMAR1CPT2CPT1A
SCHEMBL8821912 0.83 SIGMAR1 (0.49) BTKTMEM97SIGMAR1CPT2CPT1A
SCHEMBL8487974 0.81 CPT2 (0.43) BTKTMEM97SIGMAR1CPT2CPT1A
SCHEMBL8604095 0.77 BTK (0.47) BTKTMEM97SIGMAR1CPT2CPT1A
SCHEMBL8603751 0.77 BTK (0.47) BTKTMEM97SIGMAR1CPT2CPT1A
SCHEMBL8491343 0.77 BTK (0.45) BTKTMEM97SIGMAR1CPT2CPT1A
SCHEMBL8485395 0.76 BTK (0.44) BTKTMEM97SIGMAR1CPT2CPT1A
SCHEMBL8488861 0.76 BTK (0.43) BTKTMEM97SIGMAR1CPT2CPT1A
SCHEMBL8605126 0.74 BTK (0.46) BTKTMEM97SIGMAR1CPT2CPT1A
SCHEMBL8488352 0.73 BTK (0.44) BTKTMEM97SIGMAR1CPT2CPT1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5859041-A Substituted imidazoles having cytokine inhibitory activity MERCK & CO., INC. (US) 1999-01-12 US disclosed