SCHEMBL8489555

SCHEMBL8489555

Cc1cnc2c(N)cccc2c1NC(=O)Nc1ccccc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.45
RAB9A P51151 2/20 0.45
HTT P42858 1/20 0.45
ATM Q13315 1/20 0.45
KMT2A Q03164 4/20 0.43
MEN1 O00255 2/20 0.43
GBA1 P04062 1/20 0.43
SMN1; SMN2 Q16637 2/20 0.42
TP53 P04637 1/20 0.42
EPHX1 P07099 1/20 0.42
TSHR P16473 1/20 0.42
EPHX2 P34913 1/20 0.42
CDK9 P50750 1/20 0.42
CLK4 Q9HAZ1 1/20 0.42
MAPT P10636 2/20 0.42
KDM4E B2RXH2 1/20 0.42
ADORA3 P0DMS8 2/20 0.41
DDX3X O00571 1/20 0.40
ALDH1A1 P00352 1/20 0.40
TAAR1 Q96RJ0 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8488066 0.86 GCK (0.39) SMN1; SMN2KDM4EALDH1A1
SCHEMBL8489810 0.85 NPSR1 (0.45) NPC1RAB9AHTTKMT2AMEN1
SCHEMBL8489309 0.83 KDM4E (0.39) KDM4E
SCHEMBL8489156 0.82 KDM4E (0.39) KMT2AMEN1MAPTKDM4E
SCHEMBL8489999 0.82 ABL1 (0.38)
SCHEMBL8490559 0.82 LMNA (0.56) NPC1RAB9AHTTATMKMT2A
SCHEMBL8487080 0.81 EPHX1 (0.45) NPC1RAB9AEPHX1MAPT
SCHEMBL8486440 0.80 KDM4E (0.36) KDM4E
SCHEMBL8486963 0.78 MAPK1 (0.41) SMN1; SMN2KDM4EALDH1A1
SCHEMBL8486913 0.78 POLB (0.41) NPC1RAB9AKMT2AMEN1EPHX1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1999021835-A1 QUINOLINE DERIVATIVES AS H+-ATPase INHIBITORS AND AS BONE RESORPTION INHIBITORS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1999-05-06 WO disclosed