SCHEMBL8489558

SCHEMBL8489558

CC(=O)CCN1CCO[C@@H]2CN(c3c(F)cc4c(=O)c(C(=O)O)cn(C5CC5)c4c3F)C[C@@H]21

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 6/20 0.48
ALDH1A1 P00352 5/20 0.48
KDM4E B2RXH2 4/20 0.48
HPGD P15428 4/20 0.48
HSD17B10 Q99714 3/20 0.48
POLB P06746 2/20 0.48
OPRM1 P35372 2/20 0.48
PRKD3 O94806 1/20 0.48
ALOX15 P16050 1/20 0.48
CLK2 P49760 1/20 0.48
CLK4 Q9HAZ1 1/20 0.48
TDP1 Q9NUW8 1/20 0.48
CHRM2 P08172 1/20 0.47
CHRM1 P11229 1/20 0.47
OPRD1 P41143 1/20 0.47
TOP2A P11388 3/20 0.46
TOP2B Q02880 3/20 0.46
LMNA P02545 1/20 0.44
ALB P02768 1/20 0.44
HRH3 Q9Y5N1 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8489575 1.00 KCNH2 (0.48) KCNH2ALDH1A1KDM4EHPGDHSD17B10
SCHEMBL8489568 1.00 KCNH2 (0.48) KCNH2ALDH1A1KDM4EHPGDHSD17B10
SCHEMBL9570733 0.92 KCNH2 (0.49) KCNH2ALDH1A1KDM4EHPGDHSD17B10
SCHEMBL8329373 0.90 KCNH2 (0.40) KCNH2ALDH1A1KDM4EHPGDHSD17B10
SCHEMBL6213265 0.88 ALDH1A1 (0.52) KCNH2ALDH1A1KDM4EHPGDHSD17B10
SCHEMBL9570740 0.82 KCNH2 (0.40) KCNH2ALDH1A1KDM4EHPGDHSD17B10
SCHEMBL10809502 0.81 KDM4E (0.56) KCNH2ALDH1A1KDM4EHPGDHSD17B10
SCHEMBL6211468 0.81 ALDH1A1 (0.63) KCNH2ALDH1A1KDM4EHPGDHSD17B10
SCHEMBL9522855 0.80 KCNH2 (0.59) KCNH2ALDH1A1KDM4EHPGDHSD17B10
SCHEMBL9570903 0.79 KCNH2 (0.49) KCNH2ALDH1A1KDM4EHPGDHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6004956-A CHEMICAL INTERMEDIATES FOR BACTERICIDES BAYER AKTIENGESELLSCHAFT (DE) 1999-12-21 US disclosed
US-5532364-A FROM A DIHYDROPYRIDINE DERIVATIVE BAYER AKTIENGESELLSCHAFT (DE) 1996-07-02 US disclosed
US-5436334-A Enantiomerically pure 2-oxa-5,8-diazabicyclo[4.3.0]nonanes and process for their preparation BAYER AKTIENGESELLSCHAFT (DE) 1995-07-25 US disclosed