SCHEMBL8499112

SCHEMBL8499112

O=C(CCc1cccc2ncc(-c3cccc(F)c3)cc12)NCCc1ccccc1

nearest known ligand 0.53

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 2/20 0.50
TP53 P04637 2/20 0.50
CYP1A2 P05177 1/20 0.50
CYP2D6 P10635 1/20 0.50
CYP2C9 P11712 1/20 0.50
CYP2C19 P33261 1/20 0.50
THRB P10828 1/20 0.49
MTNR1A P48039 2/20 0.47
MTNR1B P49286 2/20 0.47
HPGD P15428 1/20 0.44
ALDH1A1 P00352 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
HCAR2 Q8TDS4 1/20 0.43
TBK1 Q9UHD2 1/20 0.43
LMNA P02545 2/20 0.42
POLB P06746 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8499069 0.85 GSK3A (0.48) MTNR1AMTNR1B
SCHEMBL8502970 0.83 PTGDR2 (0.51) MTNR1AMTNR1B
SCHEMBL8502204 0.82 THRB (0.51) TAAR1TP53CYP1A2CYP2D6CYP2C9
SCHEMBL8499494 0.82 THRB (0.51) TAAR1TP53CYP1A2CYP2D6CYP2C9
Hydrochloric Acid SCHEMBL8503257 0.78 MTNR1B (0.46) MTNR1AMTNR1B
SCHEMBL13854108 0.73 AXL (0.51) THRBALDH1A1LMNAPOLB
Hydrochloric Acid SCHEMBL8888121 0.70 GRIN2B (0.43)
SCHEMBL8499743 0.69 MAP4K4 (0.49)
Hydrochloric Acid SCHEMBL8503245 0.69 TLR8 (0.46)
SCHEMBL8504167 0.68 CDK8 (0.47) TP53HCAR2LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5646153-A INHIBITING ABNORMAL CELL PROLIFERATION RHONE-POULENC RORER PHARMACEUTICALS INC. (US) 1997-07-08 US claimed
US-RE36256-E ADMINISTERING ARYL-SUBSTITUTED QUINOXALINE DERIVATIVES AS ANTIPROLIFERATIVE, ANTICARCINOGENIC AND ANTITUMOR AGENTS RHONE-POULENC RORER PHARMACEUTICALS, INC. (US) 1999-07-20 US disclosed
US-5795889-A INHIBITING CELL GROWTH WITH ENZYME INHIBITORS FOR SKIN DISORDERS RHONE-POULENC RORER PHARMACEUTICALS INC. (US) 1998-08-18 US disclosed
US-5646153-A INHIBITING ABNORMAL CELL PROLIFERATION RHONE-POULENC RORER PHARMACEUTICALS INC. (US) 1997-07-08 US disclosed
US-5480883-A Bis mono- and bicyclic aryl and heteroaryl compounds which inhibit EGF and/or PDGF receptor tyrosine kinase RHONE-POULENC RORER PHARMACEUTICALS INC. (US) 1996-01-02 US disclosed