SCHEMBL8499155

SCHEMBL8499155

CCCCCCCCCCc1ccc(C2(NC(C)=O)COC(C)(C)OC2)cc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SPHK1 Q9NYA1 7/20 0.44
SPHK2 Q9NRA0 2/20 0.44
THRA P10827 3/20 0.43
THRB P10828 3/20 0.43
ALDH1A1 P00352 2/20 0.41
HAO1 Q9UJM8 1/20 0.41
ESR1 P03372 2/20 0.41
ADRA2A P08913 2/20 0.41
ADORA3 P0DMS8 2/20 0.41
TACR2 P21452 2/20 0.41
SLC6A2 P23975 2/20 0.41
SLC6A4 P31645 2/20 0.41
SLC6A3 Q01959 2/20 0.41
KDM4E B2RXH2 1/20 0.41
LMNA P02545 1/20 0.41
SHBG P04278 1/20 0.41
TP53 P04637 1/20 0.41
CYP3A4 P08684 1/20 0.41
HSPD1 P10809 1/20 0.41
ADRB3 P13945 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL177319 0.73 SPHK1 (0.43) SPHK1SPHK2THRATHRB
SCHEMBL565825 0.73 S1PR1 (0.49)
SCHEMBL15199332 0.73 LPL (0.48) THRATHRBALDH1A1ESR1ADRA2A
SCHEMBL2724637 0.71 THRA (0.40) SPHK1SPHK2THRATHRBHAO1
SCHEMBL19865977 0.71 ESR1 (0.42) ALDH1A1ESR1ADRA2AADORA3TACR2
SCHEMBL15541365 0.71 S1PR1 (0.43) SPHK1SPHK2THRATHRBALDH1A1
SCHEMBL19865982 0.70 HTR2A (0.47) SPHK1ALDH1A1ESR1ADRA2AADORA3
SCHEMBL11896093 0.70 HTR2A (0.47) SPHK1ALDH1A1ESR1ADRA2AADORA3
SCHEMBL19866153 0.70 ESR1 (0.44) THRATHRBALDH1A1ESR1ADRA2A
SCHEMBL176976 0.69 EPHX1 (0.44) SPHK1SPHK2THRATHRBALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5952316-A FOR TREATING AUTOIMMUNE DISEASES, E.G., RHEUMATIOD ARTHRITIS YOSHITOMI PHARMACEUTICAL INDUSTRIES, LTD. (JP) 1999-09-14 US disclosed
US-5719176-A 2-amino-1,3-propanediol compound and immunosuppressant YOSHITOMI PHARMACEUTICAL INDUSTRIES, LTD. (JP) 1998-02-17 US disclosed
US-5604229-A 2-amino-1,3-propanediol compound and immunosuppressant YOSHITOMI PHARMACEUTICAL INDUSTRIES, LTD. (JP) 1997-02-18 US disclosed
EP-0627406-A1 2-AMINO-1,3-PROPANEDIOL COMPOUND AND IMMUNOSUPPRESSANT YOSHITOMI PHARMACEUTICAL INDUSTRIES, LTD. (JP) 1994-12-07 EP disclosed