SCHEMBL8499161

SCHEMBL8499161

O=Cc1ccc(Oc2cccc3ccccc23)cc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 5/20 0.48
KMT2A Q03164 3/20 0.48
MEN1 O00255 2/20 0.48
L3MBTL1 Q9Y468 2/20 0.48
MITF O75030 1/20 0.48
POLB P06746 1/20 0.48
ALDH1A1 P00352 7/20 0.46
KDM4E B2RXH2 3/20 0.46
SMN1; SMN2 Q16637 2/20 0.46
MAPT P10636 3/20 0.46
HPGD P15428 2/20 0.46
NPSR1 Q6W5P4 2/20 0.46
HTT P42858 1/20 0.46
CARM1 Q86X55 1/20 0.45
PRMT6 Q96LA8 1/20 0.45
GAA P10253 3/20 0.44
TTR P02766 1/20 0.44
CYP1A2 P05177 1/20 0.44
CYP2C9 P11712 1/20 0.44
CYP2C19 P33261 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2078871 0.85 L3MBTL1 (0.54) LMNAKMT2AMEN1L3MBTL1MITF
SCHEMBL24815419 0.85 MAPT (0.49) LMNAKMT2AL3MBTL1ALDH1A1KDM4E
SCHEMBL30874097 0.85 MAPT (0.49) LMNAKMT2AL3MBTL1ALDH1A1KDM4E
SCHEMBL2537411 0.83 NPC1 (0.58) LMNAKMT2AMEN1L3MBTL1MITF
SCHEMBL8311249 0.83 TTR (0.58) LMNAKMT2AL3MBTL1ALDH1A1KDM4E
SCHEMBL28553442 0.83 MEN1 (0.45) LMNAKMT2AMEN1L3MBTL1MITF
SCHEMBL7538576 0.82 MAPT (0.55) LMNAL3MBTL1POLBALDH1A1KDM4E
SCHEMBL28902999 0.82 TTR (0.55) LMNAKMT2AMEN1L3MBTL1MITF
SCHEMBL10331750 0.82 ALDH5A1 (0.42) LMNAKMT2AMEN1L3MBTL1MITF
SCHEMBL10331748 0.80 ESR1 (0.44) LMNAKMT2AMEN1POLBALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0677039-B1 CYCLOBUTANE DERIVATIVES AS INHIBITORS OF SQUALENE SYNTHETASE AND PROTEIN FARNESYLTRANSFERASE ABBOTT LAB (US) 1999-03-10 EP disclosed
US-5783593-A FUNGICIDE; ANTICHOLESTEROL AGENT ABBOTT LABORATORIES (US) 1998-07-21 US disclosed
WO-1996034850-A1 CYCLOBUTANE DERIVATIVES AND THEIR USE AS INHIBITORS OF PROTEIN FARNESYLTRANSFERASE ABBOTT LABORATORIES (US) 1996-11-07 WO disclosed
EP-0677039-A1 CYCLOBUTANE DERIVATIVES AS INHIBITORS OF SQUALENE SYNTHETASE AND PROTEIN FARNESYLTRANSFERASE Abbott Laboratories (US) 1995-10-18 EP disclosed
WO-1995012572-A1 CYCLOBUTANE DERIVATIVES AS INHIBITORS OF SQUALENE SYNTHETASE AND PROTEIN FARNESYLTRANSFERASE ABBOTT LABORATORIES (US) 1995-05-11 WO disclosed