SCHEMBL8499334

SCHEMBL8499334

CCC(C(=O)O)c1ccc(Oc2c(-c3ccc(O)cc3)ccc3cc(O)ccc23)cc1

nearest known ligand 0.51

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 12/20 0.51
ESR2 Q92731 11/20 0.51
AKR1C3 P42330 7/20 0.47
AKR1C2 P52895 7/20 0.47
AKR1C1 Q04828 1/20 0.46
PTGS1 P23219 1/20 0.46
CYP2C9 P11712 1/20 0.42
HSD17B10 Q99714 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8498098 0.95 AKR1C3 (0.53) ESR1ESR2AKR1C3AKR1C2AKR1C1
SCHEMBL8502302 0.91 ESR1 (0.53) ESR1ESR2AKR1C3AKR1C2AKR1C1
SCHEMBL8497880 0.87 AKR1C3 (0.61) ESR1ESR2AKR1C3AKR1C2AKR1C1
SCHEMBL8499781 0.86 ESR1 (0.51) ESR1ESR2AKR1C3AKR1C2PTGS1
SCHEMBL8497551 0.81 APP (0.54) ESR1ESR2AKR1C3AKR1C2PTGS1
SCHEMBL8501285 0.81 ESR1 (0.48) ESR1ESR2
SCHEMBL8499778 0.80 ESR1 (0.54) ESR1ESR2
SCHEMBL8500226 0.80 ESR1 (0.46) ESR1ESR2AKR1C3AKR1C2PTGS1
SCHEMBL8497872 0.80 ESR1 (0.54) ESR1ESR2AKR1C3AKR1C2AKR1C1
SCHEMBL8499330 0.79 ESR1 (0.53) ESR1ESR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5916916-A USEFUL AS SELECTIVE ESTROGEN RECEPTOR MODULATORS. ELI LILLY AND COMPANY (US) 1999-06-29 US claimed
US-5916916-A USEFUL AS SELECTIVE ESTROGEN RECEPTOR MODULATORS. ELI LILLY AND COMPANY (US) 1999-06-29 US disclosed