SCHEMBL8501028

SCHEMBL8501028

CCC(=O)Oc1ccc(Oc2c(-c3cccc(O)c3)ccc3cc(O)ccc23)cc1

nearest known ligand 0.56

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 19/20 0.56
ESR2 Q92731 19/20 0.56
CYP1A2 P05177 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2D6 P10635 1/20 0.39
CYP2C9 P11712 1/20 0.39
HSD17B1 P14061 1/20 0.39
CYP2B6 P20813 1/20 0.39
CYP2C19 P33261 1/20 0.39
HSD17B2 P37059 1/20 0.39
THRA P10827 1/20 0.39
THRB P10828 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8497702 0.93 ESR1 (0.49) ESR1ESR2CYP1A2CYP3A4CYP2D6
SCHEMBL8502300 0.93 ESR1 (0.56) ESR1ESR2CYP1A2CYP3A4CYP2D6
SCHEMBL8498071 0.92 ESR1 (0.60) ESR1ESR2
SCHEMBL8500568 0.92 ESR1 (0.48) ESR1ESR2THRATHRB
SCHEMBL8500292 0.91 ESR1 (0.47) ESR1ESR2HSD17B1HSD17B2THRA
SCHEMBL8499778 0.90 ESR1 (0.54) ESR1ESR2
SCHEMBL8497550 0.87 ESR1 (0.49) ESR1ESR2CYP3A4CYP2D6CYP2C9
SCHEMBL8501397 0.86 ESR1 (0.54) ESR1ESR2CYP1A2CYP3A4CYP2D6
SCHEMBL8500225 0.86 ESR1 (0.48) ESR1ESR2
SCHEMBL8497867 0.86 ESR1 (0.57) ESR1ESR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5916916-A USEFUL AS SELECTIVE ESTROGEN RECEPTOR MODULATORS. ELI LILLY AND COMPANY (US) 1999-06-29 US claimed
US-5916916-A USEFUL AS SELECTIVE ESTROGEN RECEPTOR MODULATORS. ELI LILLY AND COMPANY (US) 1999-06-29 US disclosed