SCHEMBL8501397

SCHEMBL8501397

C=CCC(=O)Oc1ccc(Oc2c(-c3cccc(O)c3)ccc3cc(O)ccc23)cc1

nearest known ligand 0.54

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 19/20 0.54
ESR2 Q92731 19/20 0.54
THRA P10827 1/20 0.37
THRB P10828 1/20 0.37
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2D6 P10635 1/20 0.36
CYP2C9 P11712 1/20 0.36
HSD17B1 P14061 1/20 0.36
CYP2B6 P20813 1/20 0.36
CYP2C19 P33261 1/20 0.36
HSD17B2 P37059 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8497565 0.93 ESR1 (0.46) ESR1ESR2
SCHEMBL8501283 0.91 ESR1 (0.52) ESR1ESR2
SCHEMBL8497260 0.87 ESR1 (0.55) ESR1ESR2
SCHEMBL8498114 0.87 ESR1 (0.46) ESR1ESR2CYP3A4CYP2D6CYP2C9
SCHEMBL8501028 0.86 ESR1 (0.56) ESR1ESR2THRATHRBCYP1A2
SCHEMBL8502300 0.85 ESR1 (0.56) ESR1ESR2THRATHRBCYP1A2
SCHEMBL8500300 0.85 CYP1A2 (0.40) ESR1ESR2THRATHRBCYP1A2
SCHEMBL8500428 0.83 ESR1 (0.41) ESR1ESR2
SCHEMBL14615054 0.82 ESR1 (0.65) ESR1ESR2CYP1A2CYP3A4CYP2D6
SCHEMBL8499724 0.82 ESR1 (0.45) ESR1ESR2CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5916916-A USEFUL AS SELECTIVE ESTROGEN RECEPTOR MODULATORS. ELI LILLY AND COMPANY (US) 1999-06-29 US claimed
US-5916916-A USEFUL AS SELECTIVE ESTROGEN RECEPTOR MODULATORS. ELI LILLY AND COMPANY (US) 1999-06-29 US disclosed