SCHEMBL8501108

SCHEMBL8501108

C=CCN(C(=O)OC(C)(C)C)C(COCc1ccccc1)c1ccccc1

nearest known ligand 0.51

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 1/20 0.51
L3MBTL1 Q9Y468 4/20 0.46
PPARA Q07869 2/20 0.43
CTSS P25774 1/20 0.41
NR1H2 P55055 1/20 0.41
NR1H3 Q13133 1/20 0.41
BACE1 P56817 2/20 0.40
TACR1 P25103 3/20 0.40
PPARG P37231 1/20 0.40
MAPT P10636 1/20 0.37
MMP9 P14780 1/20 0.36
MMP14 P50281 1/20 0.36
CA1 P00915 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8502030 0.90 NPSR1 (0.47) NPSR1L3MBTL1PPARACTSSNR1H2
SCHEMBL8936940 0.88 TACR1 (0.57) TACR1
SCHEMBL27422195 0.85 NPSR1 (0.62) NPSR1L3MBTL1PPARACTSSPPARG
SCHEMBL30836091 0.84 NPSR1 (0.51) NPSR1L3MBTL1PPARACTSSPPARG
SCHEMBL24325920 0.83 SMN1; SMN2 (0.44) NPSR1L3MBTL1CTSSBACE1MAPT
SCHEMBL30836074 0.83 NPSR1 (0.50) NPSR1L3MBTL1PPARACTSSPPARG
SCHEMBL30836087 0.83 NPSR1 (0.49) NPSR1L3MBTL1PPARACTSSPPARG
SCHEMBL30836084 0.80 NPSR1 (0.47) NPSR1L3MBTL1PPARACTSSPPARG
SCHEMBL30987151 0.78 NPSR1 (0.51) NPSR1L3MBTL1PPARACTSSBACE1
SCHEMBL948156 0.75 L3MBTL1 (0.43) NPSR1L3MBTL1CTSSMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5864045-A Heterocyclic substituted piperazinone derivatives HOECHST MARION ROUSSEL, INC. (US) 1999-01-26 US disclosed
US-5840726-A Heterocyclic substituted piperazinone derivatives HOECHST MARION ROUSSEL INC. (US) 1998-11-24 US disclosed