SCHEMBL8501375

SCHEMBL8501375

C=CC(C(=O)O)c1ccc(Oc2c(-c3ccc(OC)cc3)ccc3ccccc23)cc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PPARG P37231 6/20 0.41
PPARA Q07869 6/20 0.41
GPR84 Q9NQS5 1/20 0.40
APP P05067 1/20 0.40
CYP2C19 P33261 1/20 0.40
ESR1 P03372 1/20 0.39
ESR2 Q92731 1/20 0.39
ABCG2 Q9UNQ0 1/20 0.38
MEN1 O00255 3/20 0.38
KMT2A Q03164 3/20 0.38
KDM4E B2RXH2 2/20 0.38
GLA P06280 2/20 0.38
GAA P10253 2/20 0.38
ALDH1A1 P00352 1/20 0.38
MAPT P10636 1/20 0.38
HSP90AA1 P07900 1/20 0.37
HSP90AB1 P08238 1/20 0.37
BACE1 P56817 1/20 0.37
MCL1 Q07820 1/20 0.36
MMP3 P08254 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8500430 0.91 PPARG (0.39) PPARGPPARAGPR84CYP2C19ESR1
SCHEMBL8501044 0.90 AKR1C3 (0.43) APPCYP2C19ESR1ESR2KDM4E
SCHEMBL8500328 0.89 AKR1C3 (0.42) APPCYP2C19ESR1ESR2MEN1
SCHEMBL8499017 0.88 AKR1C3 (0.39) PPARGPPARAMEN1KMT2AKDM4E
SCHEMBL8498119 0.87 ESR1 (0.43) APPCYP2C19ESR1ESR2MEN1
SCHEMBL8497557 0.85 APP (0.54) PPARGPPARAGPR84APPCYP2C19
SCHEMBL8501228 0.84 AKR1C3 (0.44) APPCYP2C19ESR1ESR2KDM4E
SCHEMBL8500221 0.84 MCL1 (0.35) PPARGPPARAESR2ABCG2MCL1
SCHEMBL8500302 0.83 AKR1C3 (0.45) GPR84CYP2C19
SCHEMBL8499729 0.83 ESR1 (0.42) PPARGPPARAESR1ESR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5916916-A USEFUL AS SELECTIVE ESTROGEN RECEPTOR MODULATORS. ELI LILLY AND COMPANY (US) 1999-06-29 US claimed
US-5916916-A USEFUL AS SELECTIVE ESTROGEN RECEPTOR MODULATORS. ELI LILLY AND COMPANY (US) 1999-06-29 US disclosed