SCHEMBL8499017

SCHEMBL8499017

C=CC(C(=O)O)c1ccc(Oc2c(-c3ccc(OC)c(Cl)c3)ccc3ccccc23)cc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKR1C3 P42330 3/20 0.39
AKR1C2 P52895 3/20 0.39
ALDH1A1 P00352 2/20 0.38
KDM4E B2RXH2 1/20 0.38
NPBWR1 P48145 3/20 0.37
ERN1 O75460 1/20 0.37
PTGS2 P35354 2/20 0.36
PTGS1 P23219 1/20 0.36
ADORA2A P29274 1/20 0.36
ADORA1 P30542 1/20 0.36
LMNA P02545 1/20 0.35
MAOB P27338 1/20 0.35
MEN1 O00255 1/20 0.35
NPC1 O15118 1/20 0.35
RAB9A P51151 1/20 0.35
KMT2A Q03164 1/20 0.35
STK39 Q9UEW8 1/20 0.35
KMO O15229 1/20 0.35
PPARG P37231 2/20 0.34
PPARA Q07869 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8500221 0.88 MCL1 (0.35) AKR1C3AKR1C2PPARGPPARA
SCHEMBL8501375 0.88 PPARG (0.41) ALDH1A1KDM4ENPBWR1MEN1KMT2A
SCHEMBL8500430 0.83 PPARG (0.39) AKR1C3AKR1C2KMT2APPARGPPARA
SCHEMBL8499012 0.83 NPBWR1 (0.40) ALDH1A1KDM4ENPBWR1ERN1PTGS2
SCHEMBL8496759 0.82 ALDH1A1 (0.39) AKR1C3ALDH1A1KDM4ENPBWR1ERN1
SCHEMBL7182545 0.81 ESR1 (0.52) ALDH1A1KDM4E
SCHEMBL7182554 0.81 ESR1 (0.52) ALDH1A1KDM4E
SCHEMBL8499729 0.81 ESR1 (0.42) AKR1C3AKR1C2PPARGPPARA
SCHEMBL8500328 0.81 AKR1C3 (0.42) AKR1C3AKR1C2ALDH1A1KDM4EPTGS2
SCHEMBL7184010 0.80 ESR1 (0.43) ALDH1A1KDM4ENPBWR1ERN1PTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5916916-A USEFUL AS SELECTIVE ESTROGEN RECEPTOR MODULATORS. ELI LILLY AND COMPANY (US) 1999-06-29 US claimed
US-5916916-A USEFUL AS SELECTIVE ESTROGEN RECEPTOR MODULATORS. ELI LILLY AND COMPANY (US) 1999-06-29 US disclosed