SCHEMBL8499729

SCHEMBL8499729

C=CC(C(=O)O)c1ccc(Oc2c(-c3cccc(F)c3)ccc3ccccc23)cc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 5/20 0.42
ESR2 Q92731 4/20 0.42
AKR1C3 P42330 5/20 0.38
AKR1C2 P52895 5/20 0.38
PPARG P37231 5/20 0.34
PPARA Q07869 4/20 0.34
TUBB4A P04350 1/20 0.34
TUBB P07437 1/20 0.34
TUBA3C P0DPH7 1/20 0.34
TUBA1B P68363 1/20 0.34
TUBA4A P68366 1/20 0.34
TUBB4B P68371 1/20 0.34
TUBB3 Q13509 1/20 0.34
TUBB2A Q13885 1/20 0.34
TUBB8 Q3ZCM7 1/20 0.34
TUBA3E Q6PEY2 1/20 0.34
TUBA1A Q71U36 1/20 0.34
TUBA1C Q9BQE3 1/20 0.34
TUBB6 Q9BUF5 1/20 0.34
TUBB2B Q9BVA1 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8500430 0.84 PPARG (0.39) ESR1ESR2AKR1C3AKR1C2PPARG
SCHEMBL8500221 0.83 MCL1 (0.35) ESR2AKR1C3AKR1C2PPARGPPARA
SCHEMBL8501375 0.83 PPARG (0.41) ESR1ESR2PPARGPPARA
SCHEMBL8501398 0.81 ESR1 (0.51) ESR1ESR2AKR1C3AKR1C2CYP1A2
SCHEMBL8499017 0.81 AKR1C3 (0.39) AKR1C3AKR1C2PPARGPPARA
SCHEMBL8497567 0.81 ESR1 (0.43) ESR1ESR2
SCHEMBL8500302 0.80 AKR1C3 (0.45) AKR1C3AKR1C2CYP1A2
SCHEMBL8500328 0.80 AKR1C3 (0.42) ESR1ESR2AKR1C3AKR1C2CYP1A2
SCHEMBL8499724 0.80 ESR1 (0.45) ESR1ESR2PPARGTUBB4ATUBB
SCHEMBL8497265 0.78 ESR1 (0.52) ESR1ESR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5916916-A USEFUL AS SELECTIVE ESTROGEN RECEPTOR MODULATORS. ELI LILLY AND COMPANY (US) 1999-06-29 US claimed
US-5916916-A USEFUL AS SELECTIVE ESTROGEN RECEPTOR MODULATORS. ELI LILLY AND COMPANY (US) 1999-06-29 US disclosed