SCHEMBL8501283

SCHEMBL8501283

C=CCC(=O)Oc1ccc(Oc2c(-c3ccc(O)cc3)ccc3cc(O)ccc23)cc1

nearest known ligand 0.52

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 19/20 0.52
ESR2 Q92731 15/20 0.52
ALDH2 P05091 1/20 0.37
MAOA P21397 1/20 0.37
MAOB P27338 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8498114 0.94 ESR1 (0.46) ESR1ESR2MAOAMAOB
SCHEMBL8497260 0.94 ESR1 (0.55) ESR1ESR2
SCHEMBL8497565 0.94 ESR1 (0.46) ESR1ESR2
SCHEMBL8501397 0.91 ESR1 (0.54) ESR1ESR2
SCHEMBL8500428 0.90 ESR1 (0.41) ESR1ESR2
SCHEMBL8501042 0.86 ESR1 (0.40) ESR1ESR2
SCHEMBL8499778 0.85 ESR1 (0.54) ESR1ESR2
SCHEMBL8499330 0.84 ESR1 (0.53) ESR1ESR2
SCHEMBL7189521 0.83 ESR1 (0.46) ESR1ESR2
SCHEMBL8501225 0.83 ESR1 (0.43) ESR1ESR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5916916-A USEFUL AS SELECTIVE ESTROGEN RECEPTOR MODULATORS. ELI LILLY AND COMPANY (US) 1999-06-29 US claimed
US-5916916-A USEFUL AS SELECTIVE ESTROGEN RECEPTOR MODULATORS. ELI LILLY AND COMPANY (US) 1999-06-29 US disclosed