SCHEMBL8501439

SCHEMBL8501439

CC(C)[C@H](NC(=O)c1cc2ccccc2n1C)C(=O)C(F)C(=O)C(N)CC(=O)O

nearest known ligand 0.55

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
TRPA1 O75762 1/20 0.51
PHGDH O43175 5/20 0.48
CNR2 P34972 3/20 0.47
MCL1 Q07820 1/20 0.43
CTSL P07711 1/20 0.42
CTSS P25774 1/20 0.42
MEN1 O00255 3/20 0.41
KMT2A Q03164 3/20 0.41
NPC1 O15118 1/20 0.41
RAB9A P51151 1/20 0.41
HDAC1 Q13547 2/20 0.41
HDAC2 Q92769 1/20 0.41
HDAC3 O15379 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8498375 0.89 MEN1 (0.51) TRPA1PHGDHMEN1KMT2AHDAC1
SCHEMBL7387717 0.89 CNR2 (0.50) TRPA1PHGDHCNR2MEN1KMT2A
SCHEMBL7390177 0.89 CNR2 (0.43) TRPA1PHGDHCNR2
SCHEMBL8525883 0.88 MEN1 (0.43) TRPA1PHGDHCNR2CTSLCTSS
SCHEMBL7390779 0.86 CNR2 (0.54) TRPA1CNR2
SCHEMBL7387933 0.85 TRPA1 (0.49) TRPA1PHGDHCNR2MCL1CTSL
SCHEMBL7390761 0.80 KDM4E (0.42) CNR2
SCHEMBL7389876 0.79 PTGER4 (0.37) CNR2MEN1KMT2ANPC1RAB9A
SCHEMBL2363959 0.79 PHGDH (0.57) TRPA1PHGDHMCL1MEN1KMT2A
SCHEMBL5667904 0.78 TRPA1 (0.50) TRPA1PHGDHCNR2MCL1CTSL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5877197-A C-terminal modified (N-substituted)-2-indolyl dipeptides as inhibitors of the ICE/ced-3 family of cysteine proteases CONATUS PHARMACEUTICALS, INC. 1999-03-02 US disclosed