SCHEMBL8501949

SCHEMBL8501949

COc1ccc(OS(=O)(=O)C(F)(F)F)cc1OC

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 3/20 0.53
CA2 P00918 3/20 0.53
CA12 O43570 3/20 0.53
CA9 Q16790 3/20 0.53
CA7 P43166 2/20 0.53
CA14 Q9ULX7 2/20 0.53
MAPK1 P28482 2/20 0.47
POLB P06746 1/20 0.47
TSHR P16473 1/20 0.47
KMT2A Q03164 2/20 0.42
MEN1 O00255 1/20 0.42
ALOX15 P16050 1/20 0.42
SMN1; SMN2 Q16637 2/20 0.42
CA4 P22748 1/20 0.42
CA6 P23280 1/20 0.42
TPMT P51580 1/20 0.42
HSD11B1 P28845 1/20 0.42
CYP1A2 P05177 1/20 0.41
CYP2C9 P11712 1/20 0.41
CYP2C19 P33261 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6938157 0.90 CA12 (0.55) CA1CA2CA12CA9CA7
SCHEMBL6935409 0.90 CA12 (0.55) CA1CA2CA12CA9CA7
SCHEMBL9710746 0.87 CA12 (0.41) CA1CA2CA12CA9CA7
SCHEMBL22444694 0.86 MAPK1 (0.47) CA1CA2MAPK1KMT2ASMN1; SMN2
SCHEMBL6360991 0.86 HSD11B1 (0.46) CA1CA2CA12CA9CA7
SCHEMBL8499142 0.85 HTR1D (0.43) CA1CA2CA12CA9CA7
SCHEMBL3125396 0.83 SMN1; SMN2 (0.42) CA1CA2SMN1; SMN2HSD11B1GAA
SCHEMBL3688422 0.83 CA1 (0.44) CA1CA2CA9HSD11B1HTR1A
SCHEMBL27958821 0.83 CA1 (0.40) CA1CA2CA12CA9CA7
SCHEMBL3198514 0.82 ALDH1A1 (0.51) KMT2AMEN1SMN1; SMN2HSD11B1CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-RE36256-E ADMINISTERING ARYL-SUBSTITUTED QUINOXALINE DERIVATIVES AS ANTIPROLIFERATIVE, ANTICARCINOGENIC AND ANTITUMOR AGENTS RHONE-POULENC RORER PHARMACEUTICALS, INC. (US) 1999-07-20 US disclosed
US-5795889-A INHIBITING CELL GROWTH WITH ENZYME INHIBITORS FOR SKIN DISORDERS RHONE-POULENC RORER PHARMACEUTICALS INC. (US) 1998-08-18 US disclosed
US-5656643-A QUINOLIN PYRIDINE DERIVATIVES; USEFUL FOR TREATING CANCER, LEKEMIA, PSORIASIS, INFLAMMATORY DISODERS, BONE DISORDERS, ATHEROSCLEROSIS AND RESTENOSIS; CONTROLLS CELLULAR REPRODUCTION RHONE-POULENC RORER PHARMACEUTICALS INC. (US) 1997-08-12 US disclosed
US-5646153-A INHIBITING ABNORMAL CELL PROLIFERATION RHONE-POULENC RORER PHARMACEUTICALS INC. (US) 1997-07-08 US disclosed
US-5480883-A Bis mono- and bicyclic aryl and heteroaryl compounds which inhibit EGF and/or PDGF receptor tyrosine kinase RHONE-POULENC RORER PHARMACEUTICALS INC. (US) 1996-01-02 US disclosed
US-5409930-A Inhibits abnoramal cell proliferation; dimethoxyquinoline/ dimethylquinoline/ quinolineoxide/ and quinoxaline derivatives RHONE-POULENC RORER PHARMACEUTICALS INC. (US) 1995-04-25 US disclosed