SCHEMBL8505153

SCHEMBL8505153

COc1ccc(-n2c(C)ccc2-c2ccccc2S(N)(=O)=O)cc1Cl

nearest known ligand 0.48

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 9/20 0.48
PTGS1 P23219 7/20 0.48
PTGER1 P34995 5/20 0.47
ALDH1A1 P00352 2/20 0.46
CYP1A2 P05177 1/20 0.46
CYP2C9 P11712 1/20 0.46
HPGD P15428 1/20 0.46
CYP2C19 P33261 1/20 0.46
MAPT P10636 2/20 0.41
ALOX15 P16050 1/20 0.41
RAB9A P51151 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
HSD17B10 Q99714 1/20 0.41
CA12 O43570 1/20 0.40
CA1 P00915 1/20 0.40
CA2 P00918 1/20 0.40
CA9 Q16790 1/20 0.40
TP53 P04637 1/20 0.39
F10 P00742 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8506105 0.87 PTGER1 (0.43) PTGS2PTGS1PTGER1F10
SCHEMBL8505457 0.86 PTGS2 (0.48) PTGS2PTGS1PTGER1ALDH1A1F10
SCHEMBL8505681 0.85 PTGER1 (0.45) PTGS2PTGS1PTGER1F10
SCHEMBL8503406 0.82 F10 (0.45) PTGS2PTGS1PTGER1ALDH1A1MAPT
SCHEMBL8503364 0.82 PTGS2 (0.48) PTGS2PTGS1ALDH1A1CYP1A2MAPT
SCHEMBL8502318 0.82 PTGER1 (0.53) PTGS2PTGS1PTGER1ALDH1A1MAPT
SCHEMBL7210291 0.79 PTGS2 (0.69) PTGS2PTGS1PTGER1ALDH1A1HPGD
SCHEMBL8504990 0.79 PTGS2 (0.49) PTGS2PTGS1PTGER1ALDH1A1HPGD
SCHEMBL8502468 0.79 PTGS2 (0.51) PTGS2PTGS1PTGER1ALDH1A1HPGD
SCHEMBL8505567 0.79 PTGS2 (0.54) PTGS2PTGS1PTGER1F10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5935990-A PYRROLYL DERIVATIVES HAVING AT POSITION 1 OR 5 A PHENYL SUBSTITUTED WITH METHYLSULFONYL OR AMINOSULFONYL; INHIBIT CYCLOOXYGENASE-2 FOR USE TREATMENT OF INFLAMMATION, AS AN ANALGESIC, OR AS AN ANTIPYRETIC G.D. SEARLE & CO. (US) 1999-08-10 US disclosed