SCHEMBL8505705

SCHEMBL8505705

CC(C)(C)NC(=O)[C@@H]1CCCCN1CC(O)C(Cc1ccccc1)NC(=O)[C@H](CC(N)=O)NC(=O)c1ccc2ccccc2c1O

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 10/20 0.62
ABCC4 O15439 2/20 0.62
ABCB11 O95342 2/20 0.62
ABCB1 P08183 2/20 0.62
TACR2 P21452 2/20 0.62
TBXAS1 P24557 2/20 0.62
OPRM1 P35372 2/20 0.62
OPRD1 P41143 2/20 0.62
OPRK1 P41145 2/20 0.62
SLC6A3 Q01959 2/20 0.62
KCNH2 Q12809 2/20 0.62
ABCG2 Q9UNQ0 2/20 0.62
ABCC3 O15438 1/20 0.62
CACNA1F O60840 1/20 0.62
HTR1A P08908 1/20 0.62
DRD2 P14416 1/20 0.62
DRD3 P35462 1/20 0.62
AVPR1A P37288 1/20 0.62
HTR2B P41595 1/20 0.62
CACNA1D Q01668 1/20 0.62

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7268418 1.00 CYP3A4 (0.62) CYP3A4ABCC4ABCB11ABCB1TACR2
SCHEMBL7267493 0.91 CYP3A4 (0.59) CYP3A4ABCC4ABCB11ABCB1TACR2
SCHEMBL7267194 0.90 CYP3A4 (0.61) CYP3A4ABCC4ABCB11ABCB1TACR2
SCHEMBL7266893 0.88 CYP3A4 (0.64) CYP3A4ABCC4ABCB11ABCB1TACR2
SCHEMBL6362281 0.86 CYP3A4 (0.82) CYP3A4ABCC4ABCB11ABCB1TACR2
SCHEMBL6362279 0.86 CYP3A4 (0.82) CYP3A4ABCC4ABCB11ABCB1TACR2
SCHEMBL7267259 0.85 CYP3A4 (0.58) CYP3A4ABCC4ABCB11ABCB1TACR2
SCHEMBL7267310 0.83 ADORA3 (0.58) CYP3A4ABCC4ABCB11ABCB1TACR2
SCHEMBL7285802 0.83 ADORA3 (0.58) CYP3A4ABCC4ABCB11ABCB1TACR2
SCHEMBL7267693 0.83 ADORA3 (0.79) CYP3A4ABCC4ABCB11ABCB1TACR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6008228-A COMPRISING A MIXTURE OF CARRIER MONOGLYCERIDES OF MEDIUM CHAIN-FATTY ACIDS HOFFMAN-LA ROCHE INC. (US) 1999-12-28 US disclosed