SCHEMBL8508741

SCHEMBL8508741

COc1ccc(C(C)(C)CN)cc1F

nearest known ligand 0.58

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KIF11 P52732 1/20 0.54
KDM1A O60341 2/20 0.41
TAAR1 Q96RJ0 1/20 0.41
RAB9A P51151 2/20 0.41
LMNA P02545 1/20 0.41
MAPK1 P28482 1/20 0.41
HTT P42858 1/20 0.41
TUBB1 Q9H4B7 4/20 0.40
KDM4E B2RXH2 1/20 0.40
ATM Q13315 1/20 0.40
CD274 Q9NZQ7 1/20 0.39
MEN1 O00255 1/20 0.38
NPC1 O15118 1/20 0.38
ALDH1A1 P00352 1/20 0.38
KMT2A Q03164 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL557886 0.84 KDM4E (0.47) KIF11TAAR1KDM4EATM
SCHEMBL31347506 0.81 GAA (0.50) KIF11TAAR1RAB9ALMNAHTT
Hydrochloric Acid SCHEMBL8508446 0.81 TAAR1 (0.42) KIF11TAAR1LMNAKDM4EATM
SCHEMBL2732542 0.80 KIF11 (0.49) KIF11KDM1ARAB9ALMNAMAPK1
SCHEMBL11280334 0.76 CYP3A4 (0.44) TAAR1KDM4EATM
SCHEMBL27800149 0.76 TSHR (0.53) TAAR1RAB9ALMNAMAPK1MEN1
SCHEMBL10667796 0.76 KIF11 (0.49) KIF11KDM1ARAB9ALMNAMAPK1
SCHEMBL13413232 0.75 KIF11 (0.46) KIF11RAB9ALMNAMAPK1HTT
Hydrochloric Acid SCHEMBL11286300 0.75 CYP3A4 (0.43) TAAR1KDM4EATM
SCHEMBL3684692 0.74 NR3C2 (0.43) KIF11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0901459-A1 CALCILYTIC COMPOUNDS NPS PHARMACEUTICALS, INC. (US) 1999-03-17 EP disclosed
WO-1997037967-A1 CALCILYTIC COMPOUNDS NPS PHARMACEUTICALS, INC. (US) 1997-10-16 WO disclosed