SCHEMBL8508973

SCHEMBL8508973

CCOC=Cc1cncc(OC(C)[C@@H]2CCCN2)c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKT1 P31749 5/20 0.42
CHRNB2 P17787 7/20 0.37
CHRNA4 P43681 5/20 0.37
CHRNB4 P30926 4/20 0.35
CHRNA3 P32297 4/20 0.35
CHRNA7 P36544 1/20 0.35
CHUK O15111 1/20 0.33
DYRK3 O43781 1/20 0.33
ROCK2 O75116 1/20 0.33
MAP4K4 O95819 1/20 0.33
PIM1 P11309 1/20 0.33
PRKACA P17612 1/20 0.33
RPS6KB1 P23443 1/20 0.33
CLK2 P49760 1/20 0.33
PRKX P51817 1/20 0.33
PRKG2 Q13237 1/20 0.33
ROCK1 Q13464 1/20 0.33
DYRK1A Q13627 1/20 0.33
PRKG1 Q13976 1/20 0.33
PKN2 Q16513 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8508803 0.82 AKT1 (0.59) AKT1CHRNB2CHRNB4CHRNA3CHUK
SCHEMBL8508800 0.82 AKT1 (0.59) AKT1CHRNB2CHRNB4CHRNA3CHUK
SCHEMBL8507102 0.82 AKT1 (0.39) AKT1CHRNB2CHRNA4CHRNB4CHRNA3
SCHEMBL8506330 0.79 AKT1 (0.39) AKT1CHRNB2CHRNA4
SCHEMBL8506327 0.79 AKT1 (0.39) AKT1CHRNB2CHRNA4
SCHEMBL6584967 0.76 AKT1 (0.60) AKT1CHRNB2CHRNB4CHRNA3CHUK
SCHEMBL6233084 0.75 CHRNB2 (0.40) CHRNB2CHRNA4CHRNB4CHRNA3
SCHEMBL7411409 0.75 CHRNB4 (0.36) CHRNB2CHRNA4CHRNB4CHRNA3
SCHEMBL7406929 0.75 CHRNB4 (0.36) CHRNB2CHRNA4CHRNB4CHRNA3
SCHEMBL4962971 0.75 CHRNB2 (0.49) CHRNB2CHRNA4CHRNB4CHRNA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0934308-A1 3-PYRIDYLOXYMETHYL HETEROCYCLIC ETHER COMPOUNDS USEFUL IN CONTROLLING CHEMICAL SYNAPTIC TRANSMISSION Abbott Laboratories (US) 1999-08-11 EP disclosed
WO-1997046554-A1 3-PYRIDYLOXYMETHYL HETEROCYCLIC ETHER COMPOUNDS USEFUL IN CONTROLLING CHEMICAL SYNAPTIC TRANSMISSION ABBOTT LABORATORIES (US) 1997-12-11 WO disclosed