SCHEMBL8509225

SCHEMBL8509225

Nc1nc(N)c(N=O)c(OCc2ccc(F)cc2)n1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
MGMT P16455 7/20 1.00
CDK2 P24941 7/20 0.74
CCNA2 P20248 6/20 0.74
CCNA1 P78396 6/20 0.74
CDK1 P06493 6/20 0.74
CCNB1 P14635 5/20 0.74
MPO P05164 2/20 0.53
MEN1 O00255 1/20 0.49
CCNB2 O95067 1/20 0.49
MTOR P42345 1/20 0.49
KMT2A Q03164 1/20 0.49
ATR Q13535 1/20 0.49
CCNB3 Q8WWL7 1/20 0.49
MAOB P27338 2/20 0.43
IDO1 P14902 1/20 0.42
AGXT P21549 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2054835 0.85 MGMT (1.00) MGMTCDK2CCNA2CCNA1CDK1
SCHEMBL14383625 0.80 MGMT (0.67) MGMTCDK2CCNA2CCNA1CDK1
SCHEMBL2100316 0.78 MGMT (0.63) MGMTCDK2CCNA2CCNA1CDK1
SCHEMBL2100311 0.77 MGMT (0.62) MGMTCDK2CCNA2CCNA1CDK1
SCHEMBL7988070 0.76 CDK2 (0.77) MGMTCDK2CCNA2CCNA1CDK1
SCHEMBL4454204 0.73 CDK2 (0.66) MGMTCDK2CCNA2CCNA1CDK1
SCHEMBL2056438 0.72 CCNA2 (0.67) MGMTCDK2CCNA2CCNA1CDK1
SCHEMBL16463323 0.71 CDK2 (0.66) MGMTCDK2CCNA2CCNA1CDK1
SCHEMBL16464209 0.70 CDK2 (0.73) MGMTCDK2CCNA2CCNA1CDK1
SCHEMBL8508184 0.69 MGMT (0.55) MGMTCDK2CCNA2CCNA1CDK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5929046-A Pyrimidine and purine derivatives and their use in treating tumour cells CANCER RESEARCH CAMPAIGN TECHNOLOGY LIMITED (GB) 1999-07-27 US disclosed