SCHEMBL8513232

SCHEMBL8513232

CCOOCCC1c2ccc(O)cc2CCN1C(=O)OC(C)(C)C

nearest known ligand 0.47

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
ESR2 Q92731 6/20 0.47
ESR1 P03372 5/20 0.43
OPRK1 P41145 1/20 0.41
GHSR Q92847 11/20 0.40
DRD2 P14416 1/20 0.39
DRD1 P21728 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30645344 0.88 ESR2 (0.51) ESR2ESR1OPRK1GHSRDRD2
SCHEMBL24528881 0.88 ESR2 (0.51) ESR2ESR1OPRK1GHSRDRD2
SCHEMBL25896285 0.85 ESR2 (0.50) ESR2ESR1OPRK1GHSRDRD2
SCHEMBL3864665 0.82 ESR2 (0.47) ESR2ESR1GHSRDRD2DRD1
SCHEMBL8523114 0.80 DRD2 (0.55) ESR2ESR1OPRK1DRD2DRD1
SCHEMBL2081445 0.78 ESR2 (0.49) ESR2ESR1GHSR
SCHEMBL31505332 0.78 ESR2 (0.56) ESR2ESR1GHSRDRD2DRD1
SCHEMBL30645355 0.78 ESR2 (0.56) ESR2ESR1GHSRDRD2DRD1
SCHEMBL24528817 0.78 ESR2 (0.56) ESR2ESR1GHSRDRD2DRD1
SCHEMBL31505408 0.78 ESR2 (0.56) ESR2ESR1GHSRDRD2DRD1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012065527-A1 COMPOUDS AND USES AS L-TYPE CALCIUM CHANNEL BLOCKER AND/OR ACETYLCHOLINESTERASE INHIBITOR THEREOF 江苏先声药物研究有限公司 (CN) 2012-05-24 WO disclosed