SCHEMBL8514004

SCHEMBL8514004

CC(C)Oc1ccc(-c2ccnc(Cl)n2)cc1C(C)C

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMO O15229 4/20 0.53
AAK1 Q2M2I8 6/20 0.43
PIK3CG P48736 3/20 0.40
MAPK8 P45983 2/20 0.40
CAMKK2 Q96RR4 2/20 0.40
GSK3B P49841 1/20 0.40
S1PR1 P21453 2/20 0.36
PIK3CA P42336 1/20 0.36
PIK3CB P42338 1/20 0.36
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
S1PR3 Q99500 1/20 0.35
CCNT1 O60563 1/20 0.35
CCNA2 P20248 1/20 0.35
CDK2 P24941 1/20 0.35
CDK9 P50750 1/20 0.35
CCNA1 P78396 1/20 0.35
CDK5 Q00535 1/20 0.35
CDK5R1 Q15078 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8510729 0.82 KMO (0.54) KMOAAK1
SCHEMBL18179501 0.80 KMO (0.42) KMOAAK1PIK3CGMAPK8CAMKK2
SCHEMBL8514773 0.75 ADRB1 (0.43) KMOS1PR1PIK3CAKMT2ACLK4
SCHEMBL3397244 0.75 MAP4K4 (0.52) KMOAAK1PIK3CGPIK3CAPIK3CB
Hydrochloric Acid SCHEMBL8514967 0.74 ADRB1 (0.42) KMOS1PR1KMT2ACLK4
SCHEMBL18036606 0.74 KMO (0.67) KMOAAK1S1PR1S1PR3
SCHEMBL12408680 0.74 MEN1 (0.61) KMOPIK3CGPIK3CAPIK3CBMEN1
SCHEMBL21508293 0.72 AAK1 (0.42) KMOAAK1S1PR1S1PR3DYRK1A
SCHEMBL17744653 0.71 KMO (0.51) KMOAAK1PIK3CGS1PR1PIK3CA
SCHEMBL1469470 0.71 MAP4K4 (0.48) KMOAAK1PIK3CGPIK3CAPIK3CB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012069852-A1 PHARMACEUTICAL COMPOUNDS AS INHIBITORS OF SPHINGOSINE KINASE ALMAC DISCOVERY LIMITED (GB) 2012-05-31 WO disclosed