SCHEMBL8514015

SCHEMBL8514015

COc1ccc(-c2cccc(C(=O)c3ccccc3)c2O)cc1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC4 P56524 1/20 0.57
HDAC2 Q92769 1/20 0.57
HDAC8 Q9BY41 1/20 0.57
ALDH1A1 P00352 4/20 0.57
SMN1; SMN2 Q16637 4/20 0.57
MAPK1 P28482 3/20 0.55
HTT P42858 3/20 0.55
CYP1A2 P05177 2/20 0.55
CYP2D6 P10635 2/20 0.55
HPGD P15428 2/20 0.55
CYP2C19 P33261 2/20 0.55
LMNA P02545 1/20 0.55
PGR P06401 1/20 0.55
SLC6A2 P23975 1/20 0.55
PDE4A P27815 1/20 0.55
HRH1 P35367 1/20 0.55
SLC6A3 Q01959 1/20 0.55
PDE4D Q08499 1/20 0.55
KDM4E B2RXH2 2/20 0.52
MAPT P10636 2/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13356437 0.88 SMN1; SMN2 (0.62) HDAC4HDAC2HDAC8ALDH1A1SMN1; SMN2
SCHEMBL28461921 0.86 ALDH1A1 (0.57) HDAC4HDAC2HDAC8ALDH1A1SMN1; SMN2
SCHEMBL29091120 0.85 HNF4A (0.61) ALDH1A1MAPK1LMNAKDM4EMAPT
SCHEMBL6034374 0.85 HNF4A (0.70) HDAC4HDAC2HDAC8ALDH1A1MAPK1
SCHEMBL7824388 0.83 SMN1; SMN2 (0.64) HDAC4HDAC2HDAC8ALDH1A1SMN1; SMN2
SCHEMBL8338154 0.82 SMN1; SMN2 (0.71) ALDH1A1SMN1; SMN2MAPK1HTTCYP1A2
SCHEMBL27779618 0.81 HDAC4 (0.58) HDAC4HDAC2HDAC8SMN1; SMN2ALOX15
SCHEMBL1148224 0.80 STAT3 (0.48) HDAC4HDAC2HDAC8ALDH1A1SMN1; SMN2
SCHEMBL19604507 0.78 SMN1; SMN2 (0.89) ALDH1A1SMN1; SMN2MAPK1HTTCYP1A2
SCHEMBL9851196 0.78 KMT2A (0.70) ALDH1A1SMN1; SMN2MAPK1HTTCYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2643837-B1 ENERGY CABLE HAVING A VOLTAGE STABILIZED THERMOPLASTIC ELECTRICALLY INSULATING LAYER PRYSMIAN SPA (IT) 2015-03-04 EP claimed
EP-2643837-A1 ENERGY CABLE HAVING A VOLTAGE STABILIZED THERMOPLASTIC ELECTRICALLY INSULATING LAYER Prysmian S.p.A. (IT) 2013-10-02 EP claimed
US-20130233604-A1 ENERGY CABLE HAVING A VOLTAGE STABILIZED THERMOPLASTIC ELECTRICALLY INSULATING LAYER PRYSMIAN S.P.A. (IT) 2013-09-12 US claimed
WO-2012069864-A1 ENERGY CABLE HAVING A VOLTAGE STABILIZED THERMOPLASTIC ELECTRICALLY INSULATING LAYER PRYSMIAN S.P.A. (IT) 2012-05-31 WO claimed
EP-2643837-B1 ENERGY CABLE HAVING A VOLTAGE STABILIZED THERMOPLASTIC ELECTRICALLY INSULATING LAYER PRYSMIAN SPA (IT) 2015-03-04 EP disclosed
EP-2643837-A1 ENERGY CABLE HAVING A VOLTAGE STABILIZED THERMOPLASTIC ELECTRICALLY INSULATING LAYER Prysmian S.p.A. (IT) 2013-10-02 EP disclosed
US-20130233604-A1 ENERGY CABLE HAVING A VOLTAGE STABILIZED THERMOPLASTIC ELECTRICALLY INSULATING LAYER PRYSMIAN S.P.A. (IT) 2013-09-12 US disclosed
WO-2012069864-A1 ENERGY CABLE HAVING A VOLTAGE STABILIZED THERMOPLASTIC ELECTRICALLY INSULATING LAYER PRYSMIAN S.P.A. (IT) 2012-05-31 WO disclosed