SCHEMBL8514438

SCHEMBL8514438

CCOOCCC1NCCc2cc(O)ccc21

nearest known ligand 0.46

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
BCHE P06276 1/20 0.44
DRD2 P14416 2/20 0.43
DRD4 P21917 2/20 0.43
KDM1A O60341 1/20 0.43
KDM4E B2RXH2 2/20 0.43
MAPT P10636 2/20 0.43
PKM P14618 1/20 0.43
GAA P10253 2/20 0.43
HTT P42858 1/20 0.43
MEN1 O00255 1/20 0.40
ABL1 P00519 1/20 0.40
ALPL P05186 1/20 0.40
KMT2A Q03164 1/20 0.40
RIN1 Q13671 1/20 0.40
CA1 P00915 1/20 0.40
CA2 P00918 1/20 0.40
CA7 P43166 1/20 0.40
CA9 Q16790 1/20 0.40
CA14 Q9ULX7 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24528952 0.84 KDM1A (0.49) BCHEDRD2DRD4KDM1AKDM4E
Bromide SCHEMBL27191476 0.82 KDM1A (0.48) BCHEDRD2DRD4KDM1AKDM4E
Bromide SCHEMBL30645337 0.82 KDM1A (0.48) BCHEDRD2DRD4KDM1AKDM4E
SCHEMBL8513919 0.77 BCHE (0.44) BCHEDRD2DRD4KDM1AKDM4E
SCHEMBL8469298 0.76 KMT2A (0.48) BCHEDRD2DRD4KDM1AKDM4E
SCHEMBL8523114 0.74 DRD2 (0.55) DRD2DRD4KDM4E
Bromide SCHEMBL9531808 0.73 KDM1A (0.47) BCHEDRD2DRD4KDM1AKDM4E
SCHEMBL10348905 0.73 DRD2 (0.60) BCHEDRD2DRD4KDM1AKDM4E
SCHEMBL10348897 0.72 BCHE (0.74) BCHEDRD2DRD4KDM1AKDM4E
SCHEMBL10349436 0.72 TBXA2R (0.74) BCHEKDM4EMAPTPKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012065527-A1 COMPOUDS AND USES AS L-TYPE CALCIUM CHANNEL BLOCKER AND/OR ACETYLCHOLINESTERASE INHIBITOR THEREOF 江苏先声药物研究有限公司 (CN) 2012-05-24 WO disclosed